1. Academic Validation
  2. Nonsteroidal progesterone receptor antagonists based on 6-thiophenehydroquinolines

Nonsteroidal progesterone receptor antagonists based on 6-thiophenehydroquinolines

  • Bioorg Med Chem Lett. 2000 Mar 6;10(5):415-8. doi: 10.1016/s0960-894x(00)00011-1.
L Zhi 1 C M Tegley B Pio S J West K B Marschke D E Mais T K Jones
Affiliations

Affiliation

Abstract

Synthesis and biological evaluation of 6-thiophene 1,2-dihydro or 1,2,3,4-tetrahydroquinoline derivatives resulted in a number of potent nonsteroidal antiprogestins.

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