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Results for "

NH2-c[X-R-L-S-X]-K-G-P-(D-1Nal)

" in MedChemExpress (MCE) Product Catalog:

3

Inhibitors & Agonists

2

Peptides

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-P3346
    NH2-c[X-R-L-S-X]-K-G-P-(D-1Nal)

    		Apelin Receptor (APJ) Cardiovascular Disease
    NH2-c[X-R-L-S-X]-K-G-P-(D-1Nal) (compound 39) is a potent APJ agonist, with a Ki of 0.6 nM. NH2-c[X-R-L-S-X]-K-G-P-(D-1Nal) can activate Gαi1 (EC50=0.8 nM) and recruit β-arrestin2 (EC50=31 nM). NH2-c[X-R-L-S-X]-K-G-P-(D-1Nal) exhibits prolonged cardiac effects [1].
    <em>NH2</em>-c[X-R-L-S-X]-K-G-P-(D-<em>1Nal</em>)
  • HY-P1432
    K-(D-1-Nal)-FwLL-NH2

    		GHSR Metabolic Disease
    K-(D-1-Nal)-FwLL-NH2 is a high affinity, potent and inverse ghrelin receptor agonist (EC50=3.4 nM, Ki=4.9 nM). K-(D-1-Nal)-FwLL-NH2 can be used for the research of obesity [1].
    K-(D-<em>1-Nal</em>)-FwLL-<em>NH2</em>
  • HY-P1432A
    K-(D-1-Nal)-FwLL-NH2 TFA

    		GHSR
    K-(D-1-Nal)-FwLL-NH2 TFA is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). K-(D-1-Nal)-FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
    K-(D-<em>1-Nal</em>)-FwLL-<em>NH2</em> TFA

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