K-(D-1-Nal)-FwLL-NH2
Based on 1 Customer Validation
K-(D-1-Nal)-FwLL-NH2 is a high affinity, potent and inverse ghrelin receptor agonist (EC50=3.4 nM, Ki=4.9 nM). K-(D-1-Nal)-FwLL-NH2 can be used for the research of obesity.
For research use only. We do not sell to patients.
- Purity : 99.56%
- CAS No.: 1394288-22-2
- Formula: C51H67N9O6
- Molecular Weight:902.13
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Storage:
Sealed storage, away from moisture.
Powder -80°C, 2 years , -20°C, 1 year* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
EC50: 3.4 nM (ghrelin receptor), Ki: 4.9 nM (ghrelin receptor)[1]
Chemical Information
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CAS No. 1394288-22-2
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Appearance Solid
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Molecular Weight 902.13
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Formula C51H67N9O6
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Color White to off-white
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Sequence
Lys-{D-Nal}-Phe-{D-Trp}-Leu-Leu-NH2
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Sequence Shortening
K-{D-Nal}-F-{D-Trp}-LL-NH2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Sealed storage, away from moisture
Powder -80°C 2 years -20°C 1 year * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Solvent & Solubility
In Vitro:
DMSO : 100 mg/mL (110.85 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (272 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.1085 mL | 5.5424 mL | 11.0849 mL | 27.7122 mL |
| 5 mM | 0.2217 mL | 1.1085 mL | 2.2170 mL | 5.5424 mL | |
| 10 mM | 0.1108 mL | 0.5542 mL | 1.1085 mL | 2.7712 mL | |
| 15 mM | 0.0739 mL | 0.3695 mL | 0.7390 mL | 1.8475 mL | |
| 20 mM | 0.0554 mL | 0.2771 mL | 0.5542 mL | 1.3856 mL | |
| 25 mM | 0.0443 mL | 0.2217 mL | 0.4434 mL | 1.1085 mL | |
| 30 mM | 0.0369 mL | 0.1847 mL | 0.3695 mL | 0.9237 mL | |
| 40 mM | 0.0277 mL | 0.1386 mL | 0.2771 mL | 0.6928 mL | |
| 50 mM | 0.0222 mL | 0.1108 mL | 0.2217 mL | 0.5542 mL | |
| 60 mM | 0.0185 mL | 0.0924 mL | 0.1847 mL | 0.4619 mL | |
| 80 mM | 0.0139 mL | 0.0693 mL | 0.1386 mL | 0.3464 mL | |
| 100 mM | 0.0111 mL | 0.0554 mL | 0.1108 mL | 0.2771 mL |
K-(D-1-Nal)-FwLL-NH2 Related Classifications
HY-P1432 Related Classifications
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