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Results for "

Trimipramine

" in MedChemExpress (MCE) Product Catalog:

5

Inhibitors & Agonists

2

Isotope-Labeled Compounds

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-B1213
    Trimipramine maleate

    		5-HT Receptor Bacterial Neurological Disease
    Trimipramine maleate is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively . Trimipramine maleate is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 μM, 2.11 μM, 3.72 μM, 8.00 μM, respectively . Trimipramine maleate has vascular activity and anxiolytic efficacy .
    <em>Trimipramine</em> maleate
  • HY-B1213A
    Trimipramine

    Trimipramine is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively. Trimipramine is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 μM, 2.11 μM, 3.72 μM, 8.00 μM, respectively. Trimipramine has vascular activity and anxiolytic efficacy .
    <em>Trimipramine</em>
  • HY-147333
    Trimipramine N-oxide

    		Drug Metabolite Neurological Disease
    Trimipramine N-oxide is an active metabolite of the tricyclic antidepressant trimipramine. Trimipramine N-oxide inhibits the human monoamine transporters for noradrenaline (hNAT), serotonin (hSERT), dopamine (hDAT) and the human organic cation transporters (hOCT1 and hOCT2) with IC50s of 11.7, 3.59, 9.4, 9.35 and 27.4 nM, respectively. Trimipramine N-oxide can be used for the research of depression and anxiety .
    <em>Trimipramine</em> N-oxide
  • HY-B1213S
    Trimipramine-d3 maleate

    		5-HT Receptor Bacterial Neurological Disease
    Trimipramine-d3 (maleate) is the deuterium labeled Trimipramine maleate. Trimipramine maleate is a 5-HT receptor antagonist, with pKis of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively[1][2].
    <em>Trimipramine</em>-d3 maleate
  • HY-B1213AS
    Trimipramine-d3 (N-methyl-d3) (maleate)

    		Bacterial 5-HT Receptor Isotope-Labeled Compounds Others
    Trimipramine-d3 (N-methyl-d3) (maleate) is the deuterium labeled Trimipramine (N-methyl) maleate[1].
    <em>Trimipramine</em>-d3 (N-methyl-d3) (maleate)

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