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NEO2734 (EP31670) is an orally active p300/CBP and BET bromodomain selective inhibitor, with IC50 values of <30 nM for both p300/CBP and BET bromodomains.
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- October 2020 (1)
- Anti-infection
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Anti-infection
Apoptosis
Cell Cycle/DNA Damage
Cytoskeleton
Epigenetics
GPCR/G Protein
- 5-HT Receptor
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Immunology/Inflammation
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
- 11β-HSD
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- 5 alpha Reductase
- Acetolactate Synthase (ALS)
- Acetyl-CoA Carboxylase
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- ACSL Family
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- Aminotransferases (Transaminases)
Neuronal Signaling
- 5-HT Receptor
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- Amino Acid Decarboxylase
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- FAAH
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PROTAC
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- E3 Ligase Ligand-Linker Conjugates
- Hsp-targeting Chimeras
- HyT
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- PROTAC-Linker Conjugates for PAC
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Protein Tyrosine Kinase/RTK
Stem Cell/Wnt
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- Recombinant Proteins
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- Cytokines and Growth Factors
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CAR-T Related Proteins
- CD4
- CD19
- CD27 Ligand/CD70
- CD123
- CD138/Syndecan-1
- Epithelial Cell Adhesion Molecule (EpCAM)
- Folate Receptor 1
- GPC-3
- Guanylate Cyclase 2C
- ErbB2/HER2
- ErbB3/HER3
- c-Met/HGFR
- MSLN
- CA-125
- ROR1
- CEACAM-5
- Prostate Specific Membrane Antigen
- TROP-2
- Siglec-6
- Folate Receptor alpha (FR-alpha)
- CD314/NKG2D
- CD319/SLAMF7
- Siglec-3/CD33
- CD7
- MUC-1/CD227
CD Antigens
- T Cell CD Proteins
- B Cell CD Proteins
- NK Cell CD Proteins
- Macrophage CD Proteins
- Monocyte CD Proteins
- Stem Cell CD Proteins
- Platelet CD Proteins
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- Dendritic Cell CD Proteins
- Epithelial cell CD Proteins
- Endothelial cell CD Proteins
- Signal Transduction-related CD Proteins
- Cell Adhesion-related CD Proteins
Receptor Proteins
- Receptor Tyrosine Kinases
- Receptor Serine/Threonine Kinases
- Receptor Tyrosine Phosphatase
- Receptor Guanylyl Cyclase Family
- Cell Adhesion Molecules (CAMs)
- G-Protein-Coupled Receptors (GPCRs)
- Nuclear Receptor Superfamily
- Pattern Recognition Receptors
- Notch family
- Siglec
- Leukocyte Immunoglobin-like Receptors
- Killer-Cell Immunoglobulin-like Receptors
- Cytokine Receptors
Enzymes & Regulators
- Oxidoreductases (EC 1)
- Transferases (EC 2)
- Hydrolases (EC 3)
- Lyases (EC 4)
- Isomerases (EC 5)
- Ligases (EC 6)
- Translocases (EC 7)
- Matrix Metalloproteinases
- ADAMs/ADAMTSs
- Cathepsin
- Carboxypeptidase
- Angiotensin-converting Enzymes
- Caspase
- Carbonic Anhydrase
- Serine/Threonine Kinase Proteins
- Protein Tyrosine Kinases
- Phosphatase
- Topoisomerase
- Protease Inhibitors
- Protein Kinase Inhibitor Peptide (PKI)
- Cyclin-Dependent Kinase Inhibitor Proteins
- Cystatin Family
- Molecular Biology
- •Nucleic Acid Gel Electrophoresis
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- Cell Biology
- •Cell Culture
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- •Cell Isolation
- View More
Cell Analysis
- Cell Proliferation and Cytotoxicity
- Reporter Gene Testing
- Phalloidin Dye Conjugates
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- AntiFade Mounting Medium
- Mitochondrial Isolation
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