1. GPCR/G Protein
    Neuronal Signaling
  2. Dopamine Receptor
    5-HT Receptor
  3. cis-(Z)-Flupentixol dihydrochloride

cis-(Z)-Flupentixol dihydrochloride (Synonyms: cis-(Z)-Flupenthixol dihydrochloride)

Cat. No.: HY-15856
Handling Instructions

cis-(Z)-Flupentixol dihydrochloride is a potent and selective DA D1/D2 receptor antagonist, with Ki values of 0.38 nM and 7 nM for D2 receptor and 5-HT2A, respectively.

For research use only. We do not sell to patients.

cis-(Z)-Flupentixol dihydrochloride Chemical Structure

cis-(Z)-Flupentixol dihydrochloride Chemical Structure

CAS No. : 51529-01-2

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Description

cis-(Z)-Flupentixol dihydrochloride is a potent and selective DA D1/D2 receptor antagonist, with Ki values of 0.38 nM and 7 nM for D2 receptor and 5-HT2A, respectively[1][2].

IC50 & Target[2]

D2 Receptor

0.38 nM (Ki)

5-HT2A Receptor

7 nM (Ki)

In Vivo

cis-(Z)-Flupentixol (0.25, or 0.5 mg/kg, i.p.) pretreatment dose-dependently reduces cocaine-induced activity[1].

Animal Model: Rats[1].
Dosage: 0.125, 0.25, or 0.5 mg/kg.
Administration: IP.
Result: Reduced cocaine-induced activity.
Molecular Weight

507.44

Formula

C₂₃H₂₇Cl₂F₃N₂OS

CAS No.

51529-01-2

SMILES

OCCN1CCN(CC/C=C2C3=C(SC4=C\2C=CC=C4)C=CC(C(F)(F)F)=C3)CC1.[H]Cl.[H]Cl

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

cis-(Z)-Flupentixolcis-(Z)-FlupenthixolDopamine Receptor5-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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cis-(Z)-Flupentixol dihydrochloride
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HY-15856
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