1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. 5-HT Receptor
  4. 5-HT Receptor Inhibitors

5-HT Receptor Inhibitors

5-HT1 Receptor

5-HT2 Receptor

5-HT3 Receptor

5-HT4 Receptor

5-HT5 Receptor

5-HT6 Receptor

5-HT7 Receptor

5-HT Receptor

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Please try each isoform separately.

5-HT Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name 5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor Purity
Puerarin  
5-HT2C Receptor
            99.42%
Clozapine  
5-HT2A Receptor, Ki: 4 nM (Inhibitor)
            99.97%
Risperidone  
5-HT2A Receptor, Ki: 4.8 nM
            99.92%
SB-699551        
5-HT5A Receptor, pKi: 8.3
     
GTS-21 dihydrochloride    
5-HT3A Receptor, IC50: 3.1 μM
          99.92%
Olanzapine
5-HT1 Receptor, Ki: 7 nM
5-HT2A Receptor, Ki: 4 nM
5-HT2C Receptor, Ki: 11 nM
5-HT3 Receptor, Ki: 57 nM
   
5-HT6 Receptor, Ki: 5 nM
    99.83%
Amitriptyline hydrochloride
5-HT1A Receptor, IC50: 450 nM
5-HT1B Receptor, IC50: 40 nM
5-HT2A Receptor, IC50: 4 nM
5-HT2B Receptor, IC50: 40 nM
5-HT2C Receptor, IC50: 6 nM
            99.28%
Aripiprazole
5-HT1A Receptor, Ki: 4.2 nM
              99.95%
Vortioxetine    
5-HT3A Receptor, Ki: 3.7 nM
     
Human 5-HT7 Receptor , Ki: 19 nM
  99.81%
Ondansetron    
5-HT3 Receptor
          99.46%
Brexpiprazole
5-HT1A Receptor, Ki: 0.12 nM
5-HT2A Receptor, Ki: 0.47 nM
            99.85%
Thioridazine hydrochloride              
serotonin
99.96%
SEP-363856 hydrochloride
5-HT1A Receptor, EC50: 2.3 μM
5-HT1B Receptor, EC50: 15.6 μM
5-HT1D Receptor, EC50: 0.262 μM
5-HT2A Receptor, EC50: >10 μM
5-HT2C Receptor, EC50: 30 μM
       
5-HT7 Receptor, EC50: 6.7 μM
  99.57%
Volinanserin  
5-HT2 Receptor, Ki: 0.36 nM
            99.76%
SB-269970 hydrochloride            
5-HT7 Receptor, pKi: 8.3
  99.15%
Cisapride      
5-HT4 Receptor, EC50: 0.14 μM
        99.72%
Ketanserin  
5-HT2 Receptor
            99.89%
Vortioxetine hydrobromide    
5-HT3A Receptor, Ki: 3.7 nM
     
5-HT7 Receptor, Ki: 19 nM
  99.91%
8-OH-DPAT
5-HT1A Receptor, pIC50: 8.19
         
5-HT7 Receptor, Ki: 466 nM
  99.26%
Tegaserod maleate  
5-HT2B Receptor (Antagonist)
 
5-HT4 Receptor (Agonist)
        99.93%
SB 242084  
5-HT2C Receptor, pKi: 9.0
            99.76%
Pimavanserin  
5-HT2A Receptor, pIC50: 8.7
            99.84%
Lurasidone
5-HT1A Receptor, IC50: 6.75 nM
         
5-HT7 Receptor, IC50: 0.495 nM
  99.90%
Vilazodone Hydrochloride
5-HT1A Receptor
              99.94%
Quetiapine
5-HT1A Receptor, pKi: 5.74
5-HT1A Receptor, pEC50: 4.77
5-HT2A Receptor, pKi: 7.54
5-HT2C Receptor, pKi: 5.55
            99.88%
Perphenazine
5-HT1A Receptor, Ki: 421 nM
5-HT2A Receptor, Ki: 5.6 nM
     
5-HT6 Receptor, Ki: 17 nM
5-HT7 Receptor, Ki: 23 nM
  99.95%
Nuciferine
5-HT1A Receptor, EC50: 3.2 μM
5-HT2C Receptor, IC50: 131 nM
5-HT2A Receptor, IC50: 478 nM
5-HT2B Receptor, IC50: 1 μM
     
5-HT6 Receptor, EC50: 700 nM
5-HT7 Receptor, IC50: 150 nM
  99.46%
Pindolol
5-HT1A Receptor
              99.91%
Agomelatine  
5-HT2C Receptor, pKi: 6.4 (native porcine)
5-HT2C Receptor, pKi: 6.2 (human)
            99.88%
Paliperidone  
5-HT2A Receptor
            99.69%
Ritanserin  
5-HT2 Receptor, IC50: 0.9 nM
            99.78%
BW-723C86  
5-HT2B Receptor
            99.80%
WAY-100635
5-HT1A Receptor, pIC50: 8.87
5-HT1A Receptor, pA2: 9.71
              99.32%
Ziprasidone
Rat 5-HT1A Receptor, Ki: 3.4 nM
human 5-HT1A Receptor, Ki: 2.5 nM
Rat 5-HT2A, Ki: 0.42 nM
            99.81%
Vilazodone
5-HT1A Receptor
              99.84%
Alprenolol hydrochloride
5-HT1A Receptor
              99.76%
GR 113808
5-HT1A Receptor
5-HT2A Receptor
5-HT2C Receptor
5-HT3 Receptor
5-HT4 Receptor
        99.96%
Sumatriptan succinate
5-HT1D Receptor, Ki: 17 nM
5-HT1B Receptor, Ki: 27 nM
5-HT1A Receptor, Ki: 100 nM
5-HT1D Receptor, IC50: 7.3 nM
5-HT1B Receptor, IC50: 9.3 nM
5-HT1F Receptor, IC50: 17.8 nM
              99.94%
Mirtazapine  
5-HT2 Receptor, pKi: 8.05
5-HT3 Receptor, pKi: 8.1
          99.94%
Prucalopride      
5-HT4A Receptor, pKi: 8.6
5-HT4B Receptor, pKi: 8.1
        99.83%
8-OH-DPAT hydrobromide
5-HT1A Receptor, pIC50: 8.19
              99.89%
Cariprazine
5-HT1A Receptor, Ki: 2.6 nM
              99.83%
Cyproheptadine hydrochloride  
5-HT2 Receptor
            99.94%
Loxapine  
human 5-HT2
            99.69%
Tandospirone
5-HT1A Receptor, Ki: 27 nM
              99.41%
Sertindole  
5-HT2A Receptor
5-HT2C Receptor
            99.75%
Methiothepin mesylate
5-HT1A Receptor, pKd: 7.10
5-HT1B Receptor, pKd: 7.28
5-HT1C Receptor, pKd: 7.56
5-HT1D Receptor, pKd: 6.99
5-HT2A Receptor, pKi: 8.50
5-HT2B Receptor, pKi: 8.68
5-HT2C Receptor, pKi: 8.35
   
5-HT5A Receptor, pKd: 7.0
5-HT5B Receptor, pKd: 7.8
5-HT6 Receptor, pKd: 8.74
5-HT7 Receptor, pKd: 8.99
  99.60%
Asenapine maleate  
5-HT2A Receptor, Ki: 0.06 nM
5-HT2C Receptor, Ki: 0.03 nM
       
5-HT7 Receptor, Ki: 0.13 nM
  99.95%
SB 204741  
human 5-HT2B Receptor, pKi: 7.1
            99.91%
Cariprazine hydrochloride
5-HT1A Receptor, Ki: 2.6 nM
              99.90%
Mosapride citrate      
5-HT4 Receptor
        99.80%
SB-224289 hydrochloride
5-HT1B Receptor
              ≥99.0%
RS-127445 hydrochloride  
5-HT2A Receptor, pKi: 6.3
5-HT2C Receptor, pKi: 6.4
5-HT2B Receptor, pKi: 9.5
5-HT3 Receptor, pKi: <6
 
5-HT5 Receptor, pKi: <6
5-HT6 Receptor, pKi: <6
    99.62%
Nefazodone hydrochloride  
5-HT2A Receptor, Ki: 5.8 nM
            99.87%
Cefaclor              
5-HT Receptor
99.61%
LP-211
5-HT1A Receptor, Ki: 188 nM
         
5-HT7 Receptor, Ki: 0.58 nM
  99.61%
Lurasidone Hydrochloride
5-HT1A Receptor, IC50: 6.75 nM
         
5-HT7 Receptor, IC50: 0.495 nM
  99.96%
Syk Inhibitor II              
serotonin, IC50: 460 nM
98.05%
SKF-83566  
5-HT2 Receptor, Ki: 11 nM
            99.86%
Paliperidone palmitate  
5-HT2A Receptor
            98.41%
R 59-022              
serotonin
99.82%
Prucalopride succinate      
5-HT4A Receptor, pKi: 8.6
5-HT4B Receptor, pKi: 8.1
        99.95%
Rotigotine
5-HT1A Receptor, Ki: 30 nM
         
5-HT7 Receptor, Ki: 86 nM
  99.98%
Palonosetron hydrochloride    
5-HT3 Receptor
          99.96%
Granisetron Hydrochloride    
5-HT3 Receptor, IC50: 17 μM
          99.90%
Quetiapine hemifumarate
5-HT1A Receptor, pKi: 5.74
5-HT1A Receptor, pEC50: 4.77
5-HT2A Receptor, pKi: 7.54
5-HT2C Receptor, pKi: 5.55
            99.94%
Ondansetron hydrochloride dihydrate    
5-HT3 Receptor
          99.03%
Sarpogrelate hydrochloride  
5-HT2A Receptor, pKi: 8.52
5-HT2B Receptor, pKi: 6.57
5-HT2C Receptor, pKi: 7.43
            99.45%
NAS-181 dimesylate
Rat 5-HT1B Receptor, IC50: 47 nM
              98.44%
Loxapine succinate  
human 5-HT2
            99.81%
Piboserod      
5-HT4 Receptor
        99.09%
Sumatriptan
5-HT1A Receptor, Ki: 100 nM
5-HT1B Receptor, Ki: 27 nM
5-HT1D Receptor, Ki: 17 nM
5-HT1D Receptor, IC50: 7.3 nM
5-HT1B Receptor, IC50: 9.3 nM
5-HT1F Receptor, IC50: 17.8 nM
              99.90%
Alosetron Hydrochloride    
5-HT3 Receptor
          99.76%
Tegaserod      
5-HT4 Receptor
        99.89%
Perospirone
5-HT1A Receptor, Ki: 2.9 nM
5-HT1 Receptor, Ki: 18 nM
5-HT2A Receptor, Ki: 0.6 nM
            99.43%
Harmine hydrochloride  
5-HT2A Receptor, Ki: 397 nM
            99.93%
UNC9994 hydrochloride
5-HT1A Receptor, Ki: 26 nM
5-HT2A Receptor, Ki: 140 nM
5-HT2B Receptor, Ki: 25 nM
5-HT2C Receptor, Ki: 512 nM
            98.83%
AS19
5-HT1A Receptor, Ki: 89.7 nM
5-HT1B Receptor, Ki: 490 nM
5-HT1D Receptor, Ki: 6.6 nM
     
5-HT5 Receptor, Ki: 98.5 nM
 
Human 5-HT7 Receptor , IC50: 0.83 nM
Human 5-HT7 Receptor , Ki: 0.6 nM
  99.85%
Oxatomide              
serotonin
99.56%
Setiptiline  
5-HT2A Receptor
5-HT2C Receptor
5-HT3 Receptor
          98.04%
Setiptiline maleate  
5-HT2A Receptor
5-HT2C Receptor
5-HT3 Receptor
          99.94%
Ansofaxine hydrochloride              
serotonin, IC50: 723 nM
99.87%
Rotundine
5-HT1A Receptor, IC50: 370 nM
              99.87%
(Z)-Thiothixene              
serotonin
99.84%
Eletriptan hydrobromide
5-HT1B Receptor, Ki: 0.92 nM
5-HT1D Receptor, Ki: 3.14 nM
              99.81%
SB 258719            
5-HT7 Receptor, pKi: 7.5
  99.04%
Asenapine
5-HT1A Receptor, pKi: 8.6
5-HT1B Receptor, pKi: 8.4
5-HT2A Receptor, pKi: 10.2
5-HT2B Receptor, pKi: 9.8
5-HT2C Receptor, pKi: 10.5
   
5-HT5 Receptor, pKi: 8.8
5-HT6 Receptor, pKi: 9.6
5-HT7 Receptor, pKi: 9.9
  99.93%
LY310762
5-HT1D Receptor, Ki: 249 nM
              98.68%
Blonanserin  
5-HT2A Receptor, Ki: 0.812 nM
5-HT2C Receptor, Ki: 26.4 nM
     
5-HT6 Receptor, Ki: 11.7 nM
    99.62%
Alverine citrate
5-HT1A Receptor, IC50: 101 nM
              99.71%
Ziprasidone hydrochloride monohydrate
Rat 5-HT1A Receptor, Ki: 3.4 nM
Rat 5-HT2A, Ki: 0.42 nM
            99.74%
Tianeptine sodium salt              
serotonin
99.90%
Gepirone
5-HT1A Receptor
              98.81%
RU 24969
5-HT1B Receptor, Ki: 0.38 nM
5-HT1A Receptor, Ki: 2.5 nM
              99.77%
Pizotifen  
5-HT2A Receptor
            98.40%
Rotigotine Hydrochloride
5-HT1A Receptor, Ki: 30 nM
         
5-HT7 Receptor, Ki: 86 nM
  99.65%
F-15599
5-HT1A Receptor, Ki: 3.4 nM
              99.82%
S1RA  
human 5-HT2B Receptor, Ki: 328 nM
            99.43%
Rizatriptan benzoate
5-HT1 Receptor
              99.94%
Xanthotoxol              
serotonin
99.75%
SB 242084 dihydrochloride  
5-HT2C Receptor, pKi: 9.0
            99.10%
Naftidrofuryl oxalate  
5-HT2 Receptor
            98.39%
Intepirdine          
5-HT6 Receptor, pKi: 9.63
    98.92%
NAN-190 hydrobromide
5-HT1 Receptor
              98.59%
Flibanserin
5-HT1A Receptor, Ki: 1 nM
5-HT2A Receptor, Ki: 49 nM
            99.54%
Iloperidone
Rat 5-HT1A Receptor, Ki: 168 nM
Rat 5-HT2 Receptor, Ki: 3.1 nM
Human 5-HT2A Receptor, Ki: 5.6 nM
Human 5-HT2C Receptor, Ki: 42.8 nM
     
Rat 5-HT6 Receptor, Ki: 42.7 μM
Rat 5-HT7 Receptor, Ki: 21.6 nM
  99.97%
Mirtazapine-d3  
5-HT2 Receptor
5-HT3 Receptor
          98.55%
WAY-181187          
5-HT6 Receptor, Ki: 2.2 nM
5-HT6 Receptor, EC50: 6.6 nM
    98.07%
SB 243213
human 5-HT1A Receptor, pKi: <5.3
human 5-HT1B Receptor, pKi: 5.5
human 5-HT1D Receptor, pKi: 6.32
human 5-HT1E Receptor, pKi: <5.4
human 5-HT1F Receptor, pKi: 5.35
Human 5-HT2C Receptor, pKi: 9.37
Human 5-HT2A Receptor, pKi: 7.01
human 5-HT2B Receptor, pKi: 7.2
     
Human 5-HT6 Receptor, pKi: 6.5
Human 5-HT7 Receptor , pKi: 5.64
  98.97%
R 59-022 hydrochloride              
serotonin
98.88%
SB-277011 hydrochloride
5-HT1D Receptor
5-HT1B Receptor
              98.54%
Dolasetron    
5-HT3 Receptor
          ≥98.0%
LY 344864
human 5-HT1F Receptor, Ki: 0.006 μM
human 5-HT1A Receptor, Ki: 0.530 μM
human 5-HT1B Receptor, Ki: 0.549 μM
human 5-HT1D Receptor, Ki: 0.575 μM
human 5-HT1E Receptor, Ki: 1.415 μM
human 5-HT2B Receptor, Ki: 1.695 μM
Human 5-HT2A Receptor, Ki: 3.499 μM
Human 5-HT3A Receptor, Ki: 3.935 mM
     
Human 5-HT7 Receptor , Ki: 4.851 μM
  98.93%
Tropisetron Hydrochloride    
5-HT3 Receptor, IC50: 70.1 nM
          99.90%
Tropisetron    
5-HT3 Receptor, IC50: 70.1 nM
          98.72%
Nelotanserin  
5-HT2A Receptor, IC50: 1.7 nM
5-HT2C Receptor, IC50: 79 nM
5-HT2B Receptor, IC50: 791 nM
            99.52%
Pumosetrag Hydrochloride    
5-HT3 Receptor
          99.77%
Befiradol hydrochloride
5-HT1A Receptor
              99.93%
Xaliproden hydrochloride
5-HT1A Receptor, IC50: 3 nM
              98.57%
GR 125743
human 5-HT1B Receptor, pKi: 8.85
human 5-HT1D Receptor, pKi: 8.31
              99.84%
Geissoschizine methyl ether
5-HT1A Receptor
              99.63%
Ecopipam hydrochloride              
5-HT Receptor, Ki: 80 nM
99.46%
A-582941 dihydrochloride    
5-HT3 Receptor, Ki: 150 nM
          99.78%
Brilaroxazine
5-HT1A Receptor, Ki: 1.5 nM
5-HT2A Receptor, Ki: 2.5 nM
5-HT2B Receptor, Ki: 0.19 nM
       
5-HT7 Receptor, Ki: 2.7 nM
  98.29%
SB 271046 Hydrochloride
5-HT1D Receptor, pKi: 6.55
5-HT1A Receptor, pKi: 6.35
5-HT1B Receptor, pKi: 6.05
5-HT1F Receptor, pKi: 5.95
5-HT1E Receptor, pKi: <4.99
5-HT2A Receptor, pKi: 5.62
5-HT2B Receptor, pKi: 5.41
Human 5-HT2C Receptor, pKi: 5.73
 
5-HT4 Receptor, pKi: 5.27
 
5-HT6 Receptor, pKi: 8.92-9.02
5-HT7 Receptor, pKi: 5.39
  99.21%
Ramosetron Hydrochloride    
5-HT3 Receptor
          99.96%
Talipexole dihydrochloride    
5-HT3 Receptor
          99.80%
LY334370
5-HT1F Receptor, Ki: 1.6 nM
              99.59%
DSP-1053
5-HT1A Receptor, Ki: 5.05 nM
              99.72%
5-HT2B antagonist-1  
5-HT2B Receptor, IC50: 33.4 nM
            99.86%
3-Hydroxy agomelatine  
5-HT2C Receptor, IC50: 3.2 μM
5-HT2C Receptor, Ki: 1.8 μM
            98.00%
Eptapirone
5-HT1A Receptor
              99.91%
Velusetrag      
5-HT4 Receptor, pKi: 7.7
        99.64%
Flesinoxan
5-HT1A Receptor, EC50: 24 nM
              99.90%
Opiranserin hydrochloride  
5-HT2A Receptor, IC50: 1.3 μM
            99.44%
Dehydroaripiprazole
5-HT1A Receptor, Ki: 4.2 nM
              99.66%
p-MPPI hydrochloride
5-HT1A Receptor
              99.81%
Deramciclane  
5-HT2A Receptor
5-HT2C Receptor
            98.13%
Tetrahydro-β-carboline              
serotonin, Ki: 6.1 μM
Arotinolol  
5-HT2A Receptor
            98.23%
Valerenic acid        
5-HT5A Receptor, IC50: 17.2 μM
      ≥99.0%
Azasetron hydrochloride    
5-HT3 Receptor, IC50: 0.33 nM
          99.78%
BRL 54443
5-HT1E Receptor, Ki: 1.1 nM
5-HT1F Receptor, Ki: 0.7 nM
5-HT1A Receptor, Ki: 63 nM
5-HT1B Receptor, Ki: 126 nM
5-HT1D Receptor, Ki: 63 nM
5-HT2A Receptor, Ki: 1259 nM
5-HT2B Receptor, Ki: 100 nM
5-HT2C Receptor, Ki: 316 nM
     
5-HT6 Receptor, Ki: >10,000 nM
5-HT7 Receptor, Ki: >10,000 nM
  99.89%
Urapidil hydrochloride
5-HT1A Receptor
              99.97%
Ecopipam hydrobromide              
5-HT Receptor, Ki: 80 nM
≥99.0%
PRX-08066  
5-HT2B Receptor, IC50: 3.4 nM
           
Asenapine hydrochloride  
5-HT2A Receptor, Ki: 0.06 nM
5-HT2C Receptor, Ki: 0.03 nM
       
5-HT7 Receptor, Ki: 0.13 nM
  99.56%
Befiradol
5-HT1A Receptor
              99.74%
Piromelatine
5-HT1A Receptor (Agonist)
5-HT1D Receptor (Agonist)
5-HT2B Receptor (Antagonist)
            99.54%
Tianeptine              
serotonin
99.84%
Vabicaserin hydrochloride  
5-HT2C Receptor, EC50: 8 nM
            99.92%
Desmethyl cariprazine
5-HT1A Receptor, Ki: 2.6 nM
              98.06%
Frovatriptan succinate hydrate
5-HT1B Receptor, pEC50: 8.2
              99.60%
Fananserin  
5-HT2 Receptor, Ki: 0.37 nM
            99.97%
RS-102221 hydrochloride  
5-HT2C Receptor, Ki: 10 nM
            99.33%
LY266097 hydrochloride  
5-HT2B Receptor, pKi: 9.8
5-HT2A Receptor, pKi: 7.7
5-HT2C Receptor, pKi: 7.6
            99.60%
Norfluoxetine hydrochloride              
5-HT Receptor
99.01%
Pimethixene maleate
5-HT1A Receptor, pKi: 7.63
5-HT2A Receptor, pKi: 10.22
5-HT2B Receptor, pKi: 10.44
5-HT2C Receptor, pKi: 8.42
            99.94%
SB-399885 hydrochloride          
5-HT6 Receptor
    99.58%
BMY-14802 hydrochloride
5-HT1A Receptor
              98.02%
CP-809101 hydrochloride  
5-HT2C Receptor, pEC50: 9.96
5-HT2B Receptor, pEC50: 7.19
5-HT2A Receptor, pEC50: 6.81
            99.37%
Idalopirdine Hydrochloride          
5-HT6 Receptor, Ki: 0.83 nM
    99.96%
GSK163090
5-HT1A Receptor, pKi: 9.4
5-HT1B Receptor, pKi: 8.5
5-HT1D Receptor, pKi: 9.7
5-HT2A Receptor, pKi: 6
5-HT2B Receptor, pKi: 6.3
5-HT2C Receptor, pKi: 5.8
     
Human 5-HT6 Receptor, pKi: <5.3
Human 5-HT7 Receptor , pKi: 6.8
  99.77%
cis-Urocanic acid  
5-HT2A Receptor
            99.92%
Cinanserin hydrochloride  
5-HT2 Receptor, Ki: 41 nM
            99.48%
Masupirdine mesylate          
5-HT6 Receptor, Ki: 2.04 nM
    99.62%
Brexpiprazole S-oxide-d8
5-HT1A Receptor, Ki: 0.12 nM
5-HT2A Receptor, Ki: 0.47 nM
            98.72%
Ro60-0175  
5-HT2C Receptor
            99.98%
PRX-07034 hydrochloride
5-HT1A Receptor, Ki: 420 nM
5-HT1B Receptor, Ki: 260 nM
5-HT1D Receptor, Ki: 2.8 μM
5-HT2A Receptor, IC50: 2.5 μM
5-HT2B Receptor, IC50: 2.5 μM
5-HT2C Receptor, IC50: 3.7 μM
     
5-HT6 Receptor, Ki: 4-8 nM
5-HT6 Receptor, IC50: 19 nM
    98.09%
Agomelatine hydrochloride  
5-HT2C Receptor, pKi: 6.4 (native porcine)
5-HT2C Receptor, pKi: 6.2 (human)
            99.55%
Flumexadol  
5-HT2C Receptor, Ki: 25 nM
            99.86%
Didesmethyl cariprazine
5-HT1A Receptor
              99.79%
Cerlapirdine          
5-HT6 Receptor
    98.72%
Adoprazine
5-HT1A Receptor, pEC50: 9
5-HT1A Receptor, pKi: 9.1
         
5-HT7 Receptor, pKi: 7.2
  98.60%
Usmarapride      
5-HT4 Receptor, EC50: 44 nM
        ≥98.0%
Usmarapride free base      
5-HT4 Receptor, EC50: 44 nM
        99.91%
Ampreloxetine              
5-HT Receptor
98.49%
RS 39604      
5-HT4 Receptor, pKi: 9.1
        ≥98.0%
WAY-100135 dihydrochloride
5-HT1A Receptor, IC50: 34 nM
              ≥98.0%
Donitriptan
5-HT1B Receptor, pKi: 9.4
5-HT1D Receptor, pKi: 9.3
              98.12%
Strictosidinic acid              
5-HT Receptor
Felcisetrag      
huamn 5-HT4(c) Receptor, pKi: 9.4
        99.65%
Perospirone hydrochloride
5-HT1A Receptor, Ki: 2.9 nM
5-HT1 Receptor, Ki: 18 nM
5-HT2A Receptor, Ki: 0.6 nM
            99.94%
Indophagolin          
5-HT6 Receptor, IC50: 1.0 μM
    98.05%
Urapidil
5-HT1A Receptor
              99.30%
RS 67333 hydrochloride      
5-HT4 Receptor, pKi: 8.7
        99.73%
Naronapride      
5-HT4 Receptor
        99.79%
Org-12962  
5-HT2C Receptor, pEC50: 7.01
5-HT2A Receptor, pEC50: 6.38
5-HT2B Receptor, pEC50: 6.28
            99.93%
Spiroxatrine
5-HT1A Receptor, Ki: 3.94 nM
5-HT1B/D Receptor, Ki: 224000 nM
5-HT2 Receptor, Ki: 118.5 nM
            99.18%
ST1936  
5-HT2B Receptor, Ki: 245 nM
     
5-HT6 Receptor, Ki: 13 nM
5-HT7 Receptor, Ki: 168 nM
  99.70%
(S)-Mirtazapine  
5-HT2 Receptor
5-HT3 Receptor
          99.76%
Renzapride      
5-HT4 Receptor, Ki: 115 nM
        98.36%
Dolasetron Mesylate hydrate    
5-HT3 Receptor
          ≥99.0%
BRL-15572 dihydrochloride
5-HT1D Receptor
              99.77%
Rodatristat              
serotonin
99.11%
AVN-492          
5-HT6 Receptor, Ki: 91 pM
    99.49%
Rodatristat ethyl
5-HT1 Receptor
              ≥98.0%
Cariprazine-d6
5-HT1A Receptor, Ki: 2.6 nM
              98.00%
MAO-A/5-HT2AR-IN-1  
5-HT2A Receptor, IC50: 0.014 μM
           
Peptide 401              
serotonin
98.26%
BIMU 8      
5-HT4 Receptor, EC50: 18 nM
        ≥99.0%
SKF-83566 hydrobromide  
5-HT2 Receptor, Ki: 11 nM
           
Eplivanserin hemifumarate  
5-HT2A Receptor, IC50: 5.8 nM
5-HT2C Receptor, IC50: 120 nM
            98.07%
Viloxazine  
Human 5-HT2C Receptor, EC50: 32 μM
human 5-HT2B Receptor, IC50: 27 μM
           
SB 243213 dihydrochloride
human 5-HT1A Receptor, pKi: <5.3
human 5-HT1B Receptor, pKi: 5.5
human 5-HT1D Receptor, pKi: 6.32
human 5-HT1E Receptor, pKi: <5.4
human 5-HT1F Receptor, pKi: 5.35
Human 5-HT2C Receptor, pKi: 9.37
Human 5-HT2A Receptor, pKi: 7.01
human 5-HT2B Receptor, pKi: 7.2
     
Human 5-HT6 Receptor, pKi: 6.5
Human 5-HT7 Receptor , pKi: 5.64
  ≥99.0%
NPS ALX Compound 4a          
5-HT6 Receptor, IC50: 7.2 nM
5-HT6 Receptor, Ki: 0.2 nM
    ≥99.0%
PNU-142633
5-HT1D Receptor, Ki: 6 nM
              ≥98.0%
Fabesetron    
5-HT3 Receptor
5-HT4 Receptor
       
PF-04995274      
5-HT4 Receptor
        99.95%
Temanogrel  
5-HT2A Receptor, Ki: 4.9 nM
            98.14%
EMD 56551
5-HT1A Receptor
             
Cyamemazine  
5-HT2A Receptor, Ki: 1.5 nM
5-HT2C Receptor, Ki: 12 nM
5-HT3 Receptor, Ki: 75 nM
          99.42%
Eltoprazine hydrochloride
5-HT1A Receptor
5-HT1B Receptor
5-HT2C Receptor
            99.90%
E-3620    
5-HT3 Receptor
          98.88%
S-14506 hydrochloride
5-HT1 Receptor
5-HT2A Receptor
5-HT2C Receptor
            99.92%
Amperozide  
5-HT2A Receptor, Ki: 26 nM
            98.75%
SB 243213 hydrochloride
human 5-HT1A Receptor, pKi: <5.3
human 5-HT1B Receptor, pKi: 5.5
human 5-HT1D Receptor, pKi: 6.32
human 5-HT1E Receptor, pKi: <5.4
human 5-HT1F Receptor, pKi: 5.35
Human 5-HT2C Receptor, pKi: 9.37
Human 5-HT2A Receptor, pKi: 7.01
human 5-HT2B Receptor, pKi: 7.2
     
Human 5-HT6 Receptor, pKi: 6.5
Human 5-HT7 Receptor , pKi: 5.64
 
BMY 14802
5-HT1A Receptor
              98.96%
Iferanserin  
5-HT2A Receptor
            99.74%
OPC-14523 free base
5-HT1A Receptor, IC50: 2.3 nM
             
Repinotan
5-HT1A Receptor, Ki: 0.19 nM (In calf hippocampus)
5-HT1A Receptor, Ki: 0.25 nM (In rat and human cortex)
5-HT1A Receptor, Ki: 0.59 nM (In rat hippocampus)
         
5-HT7 Receptor, Ki: 6 nM
 
(R)-Mirtazapine    
5-HT3 Receptor
          99.79%
OPC-14523 hydrochloride
5-HT1A Receptor, IC50: 2.3 nM
              99.90%
F 13714 fumarate
5-HT1A Receptor
              98.65%
CJ033466      
5-HT4 Receptor, EC50: 9 nM
        98.29%
(Rac)-WAY-161503  
5-HT2C Receptor, Ki: 4 nM
5-HT2C Receptor, EC50: 12 nM
            ≥99.0%
Almotriptan
5-HT1B Receptor
5-HT1D Receptor
              99.94%
GR-46611
5-HT1D Receptor
              99.82%
Revexepride      
5-HT4 Receptor
        99.84%
Ro60-0175 fumarate  
5-HT2C Receptor
            99.47%
(S)-Amisulpride            
5-HT7 Receptor, Ki: 900 nM
  99.75%
SB228357  
5-HT2A Receptor, pKi: 6.9
5-HT2C Receptor, pKi: 9
5-HT2B Receptor, pKi: 8
            99.43%
SB-200646A  
5-HT2B Receptor, pKi: 7.5
5-HT2C Receptor, pKi: 6.9
5-HT2A Receptor, pKi: 5.2
            99.89%
PU02    
5-HT3A Receptor, IC50: 0.36 μM
5-HT 3 AB, IC50: 0.73 μM
          ≥99.0%
Alniditan dihydrochloride
human 5-HT1B Receptor, IC50: 1.7 nM
human 5-HT1D Receptor, IC50: 1.3 nM
5-HT1B Receptor, Kd: 0.9 nM
5-HT1D Receptor, Kd: 1.2 nM
              ≥99.0%
Tedatioxetine hydrobromide  
5-HT2A Receptor
5-HT2C Receptor
5-HT3 Receptor
          99.98%
Naluzotan
5-HT1A Receptor, IC50: 20 nM
5-HT1A Receptor, Ki: 5.1 nM
              98.05%
Velusetrag hydrochloride      
5-HT4 Receptor, pKi: 7.7
       
Aripiprazole-d8  
5-HT2A Receptor
5-HT2C Receptor
            ≥99.0%
Facinicline hydrochloride    
5-HT3 Receptor, Ki: 1.2 nM
          99.93%
Almotriptan malate
5-HT1B Receptor
5-HT1D Receptor
              99.53%
Relenopride hydrochloride  
5-HT2A Receptor, Ki: 600 nM
5-HT2B Receptor, Ki: 31 nM
5-HT2B Receptor, IC50: 2.1 μM
 
5-HT4 Receptor, Ki: 4.96 nM
        99.13%
TC-2153
5-HT1A Receptor
5-HT2A Receptor
            98.73%
(R)-Praziquantel-d11  
5-HT2B Receptor
            ≥99.0%
cis-(Z)-Flupentixol dihydrochloride  
5-HT2A Receptor, Ki: 7 nM
           
LY 344864 racemate
5-HT1F Receptor
              98.07%
Granisetron    
5-HT3 Receptor, IC50: 17 μM
          99.95%
Risperidone hydrochloride  
5-HT2 Receptor, Ki: 4.8 nM
           
(Rac)-Rotigotine hydrochloride
5-HT1A Receptor, Ki: 30 nM
5-HT2B Receptor, Ki: 27 nM
            98.66%
Alosetron    
5-HT3 Receptor
         
Mosapride      
5-HT4 Receptor
       
Isocorynoxeine  
5-HT2A Receptor, IC50: 72.4 μM
            99.97%
Eltoprazine
5-HT1A Receptor
5-HT1B Receptor
5-HT2C Receptor
           
Pimethixene
5-HT1A Receptor, pKi: 7.63
5-HT2A Receptor, pKi: 10.22
5-HT2B Receptor, pKi: 10.44
5-HT2C Receptor, pKi: 8.42
           
Ziprasidone hydrochloride
Rat 5-HT1A Receptor, Ki: 3.4 nM
Rat 5-HT2A, Ki: 0.42 nM
           
Palonosetron    
5-HT3 Receptor
         
5-HT6/7 antagonist 1  
5-HT2A Receptor
     
5-HT6 Receptor
5-HT7 Receptor
 
Lintopride    
5-HT3 Receptor
5-HT4 Receptor
       
Naratriptan
5-HT1 Receptor
             
Lesopitron dihydrochloride
5-HT1A Receptor, IC50: 125 nM (in rat hippocampal membranes)
              ≥98.0%
(±)-Fabesetron hydrochloride    
5-HT3 Receptor
5-HT4 Receptor
       
Lidanserin  
5-HT2A Receptor
            ≥98.0%
SB-269970            
Human 5-HT7 Receptor , pKi: 8.3
 
AM9405    
5-HT3 Receptor, IC50: 0.076 nM
         
Blonanserin dihydrochloride  
5-HT2A Receptor, Ki: 0.812 nM
5-HT2C Receptor, Ki: 26.4 nM
     
5-HT6 Receptor, Ki: 11.7 nM
   
UCSF648        
5-HT5A Receptor
     
SB 271046          
5-HT6 Receptor, pKi: 8.92-9.09
   
Mosapride citrate dihydrate      
5-HT4 Receptor
       
SEP-363856
5-HT1A Receptor, EC50: 2.3 μM
5-HT1B Receptor, EC50: 15.6 μM
5-HT1D Receptor, EC50: 0.262 μM
5-HT2A Receptor, EC50: >10 μM
5-HT2C Receptor, EC50: 30 μM
       
5-HT7 Receptor, EC50: 6.7 μM
 
LY334370 hydrochloride
5-HT1F Receptor, Kd: 0.446 nM
             
RU 24969 hemisuccinate
5-HT1A Receptor, Ki: 2.5 nM
5-HT1B Receptor, Ki: 0.38 nM
             
DV-7028 hydrochloride  
5-HT2 Receptor
           
CP-135807
5-HT1D Receptor, IC50: 3.1 nM (rat)
5-HT1D Receptor, IC50: 33 nM (bovine)
             
RS-102221  
5-HT2C Receptor, Ki: 10 nM
           
LY320135  
5-HT2 Receptor, Ki: 6.4 μM
           
Aripiprazole monohydrate
5-HT1A Receptor
5-HT2A Receptor
5-HT2B Receptor
5-HT2C Receptor
           
Risperidone-d6  
5-HT2A Receptor, Ki: 4.8 nM
           
U92016A hydrochloride
5-HT1A Receptor, Ki: 0.2 nM
             
WAY 163909  
5-HT2C Receptor, Ki: 10.5±1.1 nM
           
PRX933 hydrochloride  
5-HT2C Receptor
           
PRX-08066 maleate  
5-HT2B Receptor, IC50: 3.4 nM
           
GSK215083          
5-HT6 Receptor
   
Blonanserin-d5  
5-HT2 Receptor
           
SB-216641A
5-HT1B Receptor
5-HT1D Receptor
             
5-HT6/5-HT2A receptor ligand-2  
5-HT2A Receptor, Ki: 32 nM
     
5-HT6 Receptor, Ki: 25 nM
   
Robalzotan hydrochloride
5-HT1A Receptor
             
Eletriptan
5-HT1B Receptor, pKi: 8.0
5-HT1D Receptor, pKi: 8.9
             
SB-215505  
5-HT2B Receptor, pKi: 8.3
5-HT2A Receptor, pKi: 6.77
5-HT2C Receptor, pKi: 7.66
           
PNU-96415E  
5-HT2A Receptor
           
PNU-282987 free base    
5-HT3 Receptor
         
5-HT6/5-HT2A receptor ligand-1  
5-HT2A Receptor, IC50: 11 nM
     
5-HT6 Receptor, Ki: 2 nM
   
Isopteropodine  
5-HT2 Receptor
            98.66%
PF-03246799  
5-HT2C Receptor, EC50: 190 nM
5-HT2C Receptor, Ki: 160 nM
           
SB 258719 hydrochloride            
5-HT7 Receptor, pKi: 7.5
 
Dehydro Palonosetron    
5-HT3 Receptor
         
Brexpiprazole hydrochloride
5-HT1A Receptor, Ki: 0.12 nM
5-HT2A Receptor, Ki: 0.47 nM
           
Dehydroaripiprazole hydrochloride
5-HT1A Receptor, Ki: 4.2 nM
             
LY215840  
5-HT2 Receptor
       
5-HT7 Receptor
 
5-HT6/5-HT2AR antagonist-1  
5-HT2A Receptor, Ki: 39 nM
     
5-HT6 Receptor, Ki: 11 nM
   
BRL-15572 hydrochloride
5-HT1D Receptor
             
SB-221284  
5-HT2A Receptor, pKi: 6.4
5-HT2B Receptor, pKi: 7.9
5-HT2C Receptor, pKi: 8.6
           
Tandospirone hydrochloride
5-HT1A Receptor, Ki: 27 nM
             
Blonanserin-d8  
5-HT2 Receptor
           
5-HT7 receptor ligand 1            
5-HT7 Receptor, Ki: 8 nM
 
SCH-23390 maleate  
5-HT2C Receptor, Ki: 9.3 nM
           
7-Desmethyl-3-hydroxyagomelatine  
5-HT2C Receptor
           
MAO-B-IN-3          
Human 5-HT6 Receptor, Ki: 696 nM
   
WAY-181187 oxalate          
5-HT6 Receptor, Ki: 2.2 nM
5-HT6 Receptor, EC50: 6.6 nM
   
Flibanserin hydrochloride
5-HT1A Receptor, Ki: 1 nM
5-HT2A Receptor, Ki: 49 nM
           
SB399885          
5-HT6 Receptor, pKi: 9.02
Human 5-HT6 Receptor, pKi: 9.11
   
DSP-1053 benzenesulfonate
5-HT1A Receptor, Ki: 5.05 nM
             
Ecopipam              
5-HT Receptor, Ki: 80 nM
Cinitapride monotartrate
5-HT1 Receptor
5-HT2 Receptor
 
5-HT4 Receptor
       
5-HT7R antagonist 2            
5-HT7 Receptor, Ki: 67 nM
 
Asimilobine              
serotonergic receptor
5-HT2A antagonist 2  
5-HT2A Receptor, IC50: 14 nM
           
LP 12 hydrochloride
5-HT1A Receptor, IC50: 60.9 nM
5-HT2A Receptor, IC50: 1464 nM
       
5-HT7 Receptor, IC50: 0.13 nM
 
Mesulergine hydrochloride  
5-HT2C Receptor
           
WAY-181187 hydrochloride          
5-HT6 Receptor, Ki: 2.2 nM
5-HT6 Receptor, EC50: 6.6 nM
   
Bifeprunox
5-HT1A Receptor, pKi: 7.19 (cortex)
5-HT1A Receptor, pEC50: 6.37 (hippocampus)
             
5-HT6R antagonist 3
5-HT1A Receptor, Ki: 3533 nM
5-HT2A Receptor, Ki: 35 nM
     
5-HT6 Receptor, Ki: 14 nM
5-HT7 Receptor, Ki: 1449 nM
 
Eplivanserin  
5-HT2A Receptor, IC50: 5.8 nM (in rat cortical membrane)
5-HT2A Receptor, Ki: 1.14 nM
5-HT2C Receptor, IC50: 120 nM
           
EMD386088          
5-HT6 Receptor
   
Ro 04-6790          
Rat 5-HT6 Receptor, pKi: 7.26
Human 5-HT6 Receptor, pKi: 7.35
   
3-Hydroxy agomelatine-d3  
5-HT2C Receptor, IC50: 3.2 μM
5-HT2C Receptor, Ki: 1.8 μM
            99.92%
ST1936 oxalate  
5-HT2B Receptor, Ki: 245 nM
     
5-HT6 Receptor, Ki: 13 nM
Human 5-HT7 Receptor , Ki: 168 nM
 
(R)-Mirtazapine-d3    
5-HT3 Receptor
         
SB 258741 hydrochloride            
5-HT7 Receptor
 
Eplivanserin (mixture)  
5-HT2A Receptor
            99.77%
Syk Inhibitor II dihydrochloride              
5-HT Receptor, IC50: 460 nM
5-HT1A antagonist 1
5-HT1A Receptor, Ki: 35 nM
5-HT2A Receptor, Ki: 530 nM
       
5-HT7 Receptor, Ki: 462 nM
 
Ziprasidone mesylate trihydrate
Rat 5-HT1A Receptor, Ki: 3.4 nM
Rat 5-HT2 Receptor, Ki: 0.42 nM
           
AR-A 2
5-HT1A Receptor, Ki: 3070 nM
5-HT1B/D Receptor, Ki: 20 nM
5-HT2A Receptor, Ki: 339 nM
           
Sarpogrelate  
5-HT2 Receptor
           
(Rac)-WAY-161503 hydrochloride  
5-HT2C Receptor, Ki: 4 nM
5-HT2C Receptor, EC50: 12 nM
           
LY 278584    
5-HT3 Receptor, Ki: 1.62 nM
         
NAN-190
5-HT1 Receptor
             
Asenapine citrate
5-HT1A Receptor, pKi: 8.6
5-HT1B Receptor, pKi: 8.4
5-HT2A Receptor, pKi: 10.2
5-HT2B Receptor, pKi: 9.8
5-HT2C Receptor, pKi: 10.5
   
5-HT5 Receptor, pKi: 8.8
5-HT6 Receptor, pKi: 9.6
5-HT7 Receptor, pKi: 9.9
 
Mesembrine              
serotonin, Ki: 1.4 nM
S-14671
5-HT1A Receptor, pKi: 9.3
             
CART(62-76)(human,rat)              
serotonin
DR4485 hydrochloride            
5-HT7 Receptor, pKi: 8.14
 
Cisapride monohydrate      
5-HT4 Receptor, EC50: 0.14 μM
       
EMDT oxalate          
5-HT6 Receptor
   
TIK-301  
5-HT2C Receptor
5-HT2B Receptor
           
Loxapine hydrochloride  
human 5-HT2
           
AP521
5-HT1A Receptor, IC50: 94 nM (in human)
5-HT1A Receptor, IC50: 135 nM (in rat)
5-HT1B Receptor, IC50: 254 nM (in rat)
5-HT1B Receptor, IC50: 5530 nM (in human)
5-HT1D Receptor, IC50: 418 nM (in human)
     
5-HT5A Receptor, IC50: 422 nM (in human)
 
5-HT7 Receptor, IC50: 198 nM (in rat)
  98.96%
VU6067416  
5-HT2A Receptor, EC50: 189 nM
           
Urapidil-d4
5-HT1A Receptor
             
Opiranserin  
5-HT2A Receptor, IC50: 1.3 μM
           
BGC20-761  
Human 5-HT2A Receptor, Ki: 69 nM
     
Human 5-HT6 Receptor, Ki: 20 nM
   
5-HT2CR agonist 1  
5-HT2C Receptor, EC50: 121.5 nM
           
5-HT7 agonist 1            
5-HT7 Receptor
 
Antipsychotic agent-2
5-HT1A Receptor, EC50: 160 nM
5-HT2A Receptor, Kb: 96.4 nM
           
PF-4479745
5-HT1A Receptor, IC50: 500 nM
5-HT2C Receptor, EC50: 10 nM
5-HT2C Receptor, Ki: 15 nM
5-HT2A Receptor, IC50: 360 nM
5-HT2B Receptor, IC50: 67 nM
     
5-HT6 Receptor, IC50: 280 nM
   
Syk Inhibitor II dihydrochloride dihydrate              
serotonin, IC50: 460 nM
Ziprasidone mesylate
Rat 5-HT1A Receptor, Ki: 3.4 nM
Rat 5-HT2 Receptor, Ki: 0.42 nM
           
NEO 376
5-HT1 Receptor
              99.23%
Nemonapride
5-HT1A Receptor, IC50: 34 nM
             
CART(62-76)(human,rat) TFA              
serotonin
Perphenazine dihydrochloride
5-HT1A Receptor, Ki: 421 nM
5-HT2A Receptor, Ki: 5.6 nM
5-HT2C Receptor, Ki: 132 nM
     
5-HT6 Receptor, Ki: 17 nM
5-HT7 Receptor, Ki: 23 nM
 
AVN-101 hydrochloride
5-HT1A Receptor, Ki: 61 nM
5-HT1B Receptor, Ki: 720 nM
5-HT2C Receptor, Ki: 1.17 nM
5-HT2A Receptor, Ki: 1.56 nM
5-HT2B Receptor, Ki: 10.6 nM
     
5-HT6 Receptor, Ki: 2.04 nM
5-HT7 Receptor, Ki: 0.153 nM
 
LY 344864 hydrochloride
human 5-HT1F Receptor, Ki: 0.006 μM
human 5-HT1A Receptor, Ki: 0.530 μM
human 5-HT1B Receptor, Ki: 0.549 μM
human 5-HT1D Receptor, Ki: 0.575 μM
human 5-HT1E Receptor, Ki: 1.415 μM
human 5-HT2B Receptor, Ki: 1.695 μM
Human 5-HT2C Receptor, Ki: 3.499 μM
Human 5-HT3A Receptor, Ki: 3.935 μM
     
Human 5-HT7 Receptor , Ki: 4.851 μM
 
ARC 239
5-HT1A Receptor, Ki: 63.1 nM
              99.71%
Donitriptan hydrochloride
5-HT1B Receptor, pKi: 9.4
5-HT1D Receptor, pKi: 9.3
             
LE 300  
Rat 5-HT2A, pA2: 8.32
           
5-HT3 antagonist 5    
5-HT3 Receptor
          99.75%
Sumatriptan hydrochloride
5-HT1D Receptor, Ki: 17 nM
5-HT1B Receptor, Ki: 27 nM
5-HT1A Receptor, Ki: 100 nM
5-HT1D Receptor, IC50: 7.3 nM
5-HT1B Receptor, IC50: 9.3 nM
5-HT1F Receptor, IC50: 17.8 nM
             
SGS518 oxalate          
5-HT6 Receptor
   
Org-12962 hydrochloride  
5-HT2C Receptor, pEC50: 7.01
5-HT2A Receptor, pEC50: 6.38
5-HT2B Receptor, pEC50: 6.28
           
UNC9994
5-HT1F Receptor, Ki: 26 nM
5-HT2A Receptor, Ki: 140 nM
5-HT2B Receptor, Ki: 25 nM
5-HT2C Receptor, Ki: 512 nM
           
ML 10302 hydrochloride    
5-HT3 Receptor, Ki: 782 nM
5-HT4 Receptor, EC50: 4 nM
5-HT4 Receptor, Ki: 1.07 nM
       
NPS ALX Compound 4a dihydrochloride          
5-HT6 Receptor, IC50: 7.2 nM
5-HT6 Receptor, Ki: 0.2 nM
   
Frovatriptan succinate
5-HT1B Receptor, pEC50: 8.2
             
SB-200646  
5-HT2B Receptor, pKi: 7.5
5-HT2C Receptor, pKi: 6.9
5-HT2A Receptor, pKi: 5.2
           
5-HT4 antagonist 1      
5-HT4 Receptor, pKi: 9.6
        98.67%
RS 23597-190      
5-HT4 Receptor
       
Carpindolol
5-HT1B Receptor, pKd: 8.53
5-HT1D Receptor, pEC50: 5.91
5-HT1D Receptor, pKd: 6.37
             
5-HT6R/MAO-B modulator 1          
5-HT6 Receptor
   
WAY 629 hydrochloride  
5-HT2C Receptor, EC50: 426 nM
5-HT2A Receptor, EC50: 260000 nM
           
Brexpiprazole S-oxide
5-HT1A Receptor, Ki: 0.12 nM
5-HT2A Receptor, Ki: 0.47 nM
           
Masupirdine free base          
5-HT6 Receptor, Ki: 2.04 nM
   
SB-737050A          
5-HT6 Receptor
   
2-Methyl-5-HT maleate    
5-HT3 Receptor
         
F 13714
5-HT1A Receptor, pKi: 10.23
5-HT1B Receptor, pIC50: 5.12
             
Risperidone mesylate  
5-HT2A Receptor, Ki: 4.8 nM
           
Iloperidone hydrochloride
Rat 5-HT1A Receptor, Ki: 168 nM
Rat 5-HT2 Receptor, Ki: 3.1 nM
Human 5-HT2A Receptor, Ki: 5.6 nM
Human 5-HT2C Receptor, Ki: 42.8 nM
     
Rat 5-HT6 Receptor, Ki: 42.7 nM
Rat 5-HT7 Receptor, Ki: 21.6 nM
 
Agomelatine (L(+)-Tartaric acid)  
5-HT2C Receptor, pKi: 6.4 (native porcine)
5-HT2C Receptor, pKi: 6.2 (human)
            99.82%
Alosetron ((Z)-2-butenedioate)    
5-HT3 Receptor
         
Pardoprunox
5-HT1A Receptor, pEC50: 6.3
             
Dolasetron Mesylate    
5-HT3 Receptor
         
Alosetron (Hydrochloride(1:X))    
5-HT3 Receptor
         
Idalopirdine          
5-HT6 Receptor, Ki: 0.83 nM
   
Pizotifen malate  
5-HT2A Receptor
            99.88%
Piboserod hydrochloride      
5-HT4 Receptor
       
Nexopamil racemate  
5-HT2 Receptor
           
Abaperidone  
5-HT2A Receptor, IC50: 6.2 nM
           
Irindalone  
5-HT2 Receptor
           
Pancopride    
5-HT3 Receptor
         
Sulamserod      
5-HT4 Receptor
       
Alniditan
human 5-HT1B Receptor, IC50: 1.7 nM (in HEK 293 cell)
human 5-HT1D Receptor, IC50: 1.3 nM (in HEK 293 cell)
5-HT1B Receptor, Kd: 0.9 nM
5-HT1D Receptor, Kd: 1.2 nM
             
RG-12915    
5-HT3 Receptor, IC50: 0.16 nM
         
MHP 133      
5-HT4 Receptor
       
Wf-516
5-HT1A Receptor, Ki: 5 nM
5-HT2A Receptor, Ki: 40 nM
           
T 82    
5-HT3 Receptor
         
Ondansetron hydrochloride    
5-HT3 Receptor
         
CP-809101  
5-HT2C Receptor, pEC50: 9.96
5-HT2B Receptor, pEC50: 7.19
5-HT2A Receptor, pEC50: 6.81
           
Zatosetron maleate    
5-HT3 Receptor
         
(4E)-SUN9221  
5-HT2 Receptor
           
5-HT3 antagonist 1    
5-HT3 Receptor
         
5-HT3 antagonist 3    
5-HT3 Receptor, Ki: 0.25 nM
         
5-HT3-In-1    
5-HT3 Receptor
         
5-HT2 antagonist 1  
5-HT2 Receptor
           
5-HT3 antagonist 2    
5-HT3 Receptor
         
5-HT2A antagonist 1  
5-HT2A Receptor
           
5HT6-ligand-1          
5-HT6 Receptor, Ki: 1.43 nM