2. Academic Validation
  3. Bis(heteroaryl)piperazine (BHAP) reverse transcriptase inhibitors: structure-activity relationships of novel substituted indole analogues and the identification of 1-[(5-methanesulfonamido-1H-indol-2-yl)-carbonyl]-4-[3- [(1-methylethyl)amino]-pyridinyl]piperazine monomethanesulfonate (U-90152S), a second-generation clinical candidate

Bis(heteroaryl)piperazine (BHAP) reverse transcriptase inhibitors: structure-activity relationships of novel substituted indole analogues and the identification of 1-[(5-methanesulfonamido-1H-indol-2-yl)-carbonyl]-4-[3- [(1-methylethyl)amino]-pyridinyl]piperazine monomethanesulfonate (U-90152S), a second-generation clinical candidate

  • J Med Chem. 1993 May 14;36(10):1505-8. doi: 10.1021/jm00062a027.
D L Romero 1,  R A Morge,  M J Genin,  C Biles,  M Busso,  L Resnick,  I W Althaus,  F Reusser,  R C Thomas,  W G Tarpley
Affiliations

Affiliation

  • 1 Upjohn Laboratories, Kalamazoo, Michigan 49001.
PMID: 7684450 DOI: 10.1021/jm00062a027
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