2. Signaling Pathways
  3. Epigenetics
  4. Histone Demethylase
  5. KDM5 Isoform

KDM5

 

KDM5 Related Products (4):

Cat. No. Product Name Effect Purity
  • HY-102047B
    KDOAM-25 citrate
    		Inhibitor 98.11%
    KDOAM-25 citrate is a potent and highly selective histone lysine demethylases 5 (KDM5) inhibitor with IC50s of 71 nM, 19 nM, 69 nM, 69 nM for KDM5A, KDM5B, KDM5C, KDM5D, respectively.
  • HY-116761
    GSK467
    		Inhibitor 98.14%
    GSK467 is a cell penetrant and selective KDM5B (JARID1B or PLU1) inhibitor with a Ki of 10 nM and an IC50 of 26 nM.
  • HY-151483
    TK-129
    		Inhibitor
    TK-129 is an orally active, low-toxicity, potent KDM5B inhibitor (with high affinity; IC50=44 nM).
  • HY-100764
    YUKA1
    		Inhibitor 99.56%
    YUKA1 is a potent and cell permeable Lysine demethylase 5A (KDM5A) inhibitor, with an IC50 of 2.66 μM, less active on KDM5C (IC50, 7.12 μM), and is inactive on KDM5B, KDM6A or KDM6B.