2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. GABA Receptor
  4. CGP44532

CGP44532 is a GABAB receptor agonist with a pEC50 (geometric mean of the half-maximal effective concentration) value of 5.63 μM.

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CGP44532

CGP44532 화학구조

CAS No. : 133345-68-3

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CGP44532 Related Antibodies

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제품 설명

CGP44532 is a GABAB receptor agonist with a pEC50 (geometric mean of the half-maximal effective concentration) value of 5.63 μM[1].

Cellular Effect
Cell Line Type Value Description References
CHO-K1 EC50
600 nM
Compound: (R)-4
Agonist activity at human recombinant GABABreceptor expressed in CHO-K1 cells assessed as inhibition of intracellular calcium release by FLIPR
Agonist activity at human recombinant GABABreceptor expressed in CHO-K1 cells assessed as inhibition of intracellular calcium release by FLIPR
[PMID: 18578471]
Oocyte IC50
5.4 μM
Compound: R(+)-CGP-44533
Antagonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp method
Antagonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp method
[PMID: 17981464]
분자량

153.12

화학식

C4H12NO3P
CAS No.
SMILES

O=P(C)(C[C@H](O)CN)O
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
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CGP44532 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CGP44532133345-68-3CGP 44532CGP-44532GABA ReceptorGamma-aminobutyric acid Receptorγ-Aminobutyric acid Receptorantiepilepticcognitive-enhancementanalgesicantidepressantInhibitorinhibitorinhibit

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상품명:
CGP44532
Cat. No.:
HY-116197
수량:
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