2. GPCR/G Protein Neuronal Signaling
  3. Melatonin Receptor
  4. Melatonin receptor agonist 1

Melatonin receptor agonist 1 (compound 20c) is a potent melatonin receptor (MT) agonist, with Ki values of 108 nM (MT2) and 1140 nM (MT1).

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Melatonin receptor agonist 1

Melatonin receptor agonist 1 Chemical Structure

CAS No. : 2411150-76-8

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Melatonin receptor agonist 1 Related Antibodies

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Description

Melatonin receptor agonist 1 (compound 20c) is a potent melatonin receptor (MT) agonist, with Ki values of 108 nM (MT2) and 1140 nM (MT1)[1].

IC50 & Target

MT2

108 nM (Ki)

MT1

1140 nM (Ki)

In Vitro

Melatonin receptor agonist 1 (compound 20c) shows a 10 times MT2-selectivity over MT1[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Melatonin receptor agonist 1 Related Antibodies
Masse moléculaire

273.33

Formule

C15H19N3O2
CAS No.
SMILES

CCCC(NCCC1=NN=CC2=CC=C(C=C21)OC)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
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Melatonin receptor agonist 1 Related Classifications

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C1   V1   C2   V2
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    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Melatonin receptor agonist 12411150-76-8Melatonin receptor agonist1Melatonin receptor agonist-1Melatonin Receptorphthalazineagomelatineagonistmelatonin receptor (MT)G-protein coupled receptors (GPCRs)Inhibitorinhibitorinhibit

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Melatonin receptor agonist 1
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HY-147542
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