2. Membrane Transporter/Ion Channel
  3. Monoamine Transporter
  4. VMAT2-IN-4

VMAT2-IN-4 (compound 11) is a vesicular monoamine transporter-2 (VMAT2) inhibitor. VMAT2-IN-4 inhibits [3H]-DTBZ binding (Ki = 560 nM). VMAT2-IN-4 inhibits [3H]-DA (Ki = 45 nM) from entering vesicles and being taken up by cells. VMAT2-IN-4 can be used in methamphetamine addiction research.

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VMAT2-IN-4

VMAT2-IN-4 Estructura química

No. CAS : 1436695-49-6

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Descripciòn

VMAT2-IN-4 (compound 11) is a vesicular monoamine transporter-2 (VMAT2) inhibitor. VMAT2-IN-4 inhibits [3H]-DTBZ binding (Ki = 560 nM). VMAT2-IN-4 inhibits [3H]-DA (Ki = 45 nM) from entering vesicles and being taken up by cells. VMAT2-IN-4 can be used in methamphetamine addiction research[1].

IC50 & Target

VMAT2

 

Peso molecular

521.97

Fòrmula

C25H32ClF4NO4
No. CAS
SMILES

OC[C@H](O)CN1[C@@H](CCC2=CC=C(OC(F)F)C=C2)CC[C@H]1CCC3=CC=C(OC(F)F)C=C3.[H]Cl
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

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VMAT2-IN-4 Related Classifications

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  • Do most proteins show cross-species activity?

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Keywords:

VMAT2-IN-41436695-49-6Monoamine TransporterPyrrolidine analogsGZ-793ADihydrotetrabenazine binding siteN-Propane-1,2(R)-diolsInhibitorinhibitorinhibit

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Nombre del producto:
VMAT2-IN-4
Cat. No.:
HY-120788
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