SA72
SA72 is a highly selective fatty acid amide hydrolase (FAAH) inhibitor.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 934809-60-6
- Fòrmula: C21H26N2O6
- Peso molecular:402.44
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Actividad biológica
-
Chemical Information
- Pureza y Documentación
- Referencias
-
Help & FAQs
-
HY-14380
PF-3845FAAH Inhibitor -
HY-14376
RedafamdastatFAAH Inhibitor -
HY-N2365
Macamide BFAAH Inhibitor -
HY-10865
LY2183240Anandamide Uptake/FAAH Inhibitor -
HY-19740
BIA 10-2474FAAH Inhibitor -
HY-79511
FAAH-IN-2FAAH Inhibitor -
HY-10862
FAAH inhibitor 1FAAH Inhibitor -
HY-19636
JNJ-42165279FAAH Inhibitor -
HY-10864
URB-597FAAH Inhibitor -
HY-79511R
FAAH-IN-2 (Standard)FAAH Inhibitor -
HY-14376R
Redafamdastat (Standard)FAAH Inhibitor -
HY-N2365R
Macamide B (Standard)FAAH Inhibitor
Actividad biológica
Descripciòn
IC50 & Target
Fatty acid amide hydrolase (FAAH)[1]
In Vitro
Fatty acid amide hydrolase (FAAH) is the primary regulator of several bioactive lipid amides including anandamide. Inhibitors of FAAH are potentially useful for the treatment of pain, anxiety, depression, and other nervous system disorders. However, FAAH inhibitors must display selectivity for this enzyme relative to the numerous other serine hydrolases present in the human proteome in order to be therapeutically acceptable. SA-72 is also a carbamate inhibitor. However, SA-72 shows exceptional selectivity for FAAH. Tested carboxylesterases are not off-targets for SA-72. SA-72 does not have major effects on the level of carboxylesterase activities in liver microsomes[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
Chemical Information
-
No. CAS 934809-60-6
-
Peso molecular 402.44
-
Fòrmula C21H26N2O6
-
SMILES
O=C(OCC(N)=O)NCCCC1OCC(C2=C3C=CC(OC)=CC3=CC=C2)CO1
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
SA72 Related Classifications
HY-U00240 Related Classifications
Powered by Bioz