1. Signaling Pathways
  2. GPCR/G Protein
  3. Adenosine Receptor
  4. Adenosine A2B receptor (A2BR) Isoform
  5. Adenosine A2B receptor (A2BR) Antagonist

Adenosine A2B receptor (A2BR) Antagonist

Adenosine A2B receptor (A2BR) Antagonists (4):

Cat. No. Product Name Effect Purity
  • HY-103175
    Antagonist ≥99.0%
    PSB36 is a potent and selective antagonist of adenosine A1 receptor, with Kis 0.12 nM, 187 nM, 552 nM, 2300 nM, and 6500 nM for rA1, hA2B, rA2A, hA3 and rA3 receptors respectively.
  • HY-148088
    M1069 is a selective and orall active, dual A2A/A2B adenosine receptor antagonist with a selectivity of >100 fold against the A1 and A3 receptors.
  • HY-103182
    PSB-1115 is a selective A2B Adenosine Receptor antagonist.
  • HY-148076
    A2A receptor antagonist 3
    A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist with a Ki of 0.4 nM.