Cleminorexton

Cat. No.: HY-177073: Ficha de datos
SDS
Instrucciones de manejo
FAQs
Technical Support

Cleminorexton is an orally active orexin-2 receptor (OX2R) agonist with a pEC₅₀ between 9 and 10.4. Cleminorexton can be used for narcolepsy and other conditions associated with orexin deficiency and/or excessive sleepiness.

Para uso exclusivo en investigación. No vendemos a pacientes.

Cleminorexton Estructura química

No. CAS : 2980518-93-0

Tamaño	Precio	Stock
1 mg		Pide un presupuesto y un plazo de entrega
5 mg		Pide un presupuesto y un plazo de entrega

* Seleccione Cantidad antes de agregar artículos.

This product is a controlled substance and not for sale in your territory.

Recomendaciones destacadas

•Related Small Molecules:

•Related Proteins:

Ver todos los productos específicos de isoformas Orexin Receptor (OX Receptor):

Ver todas las isoformas

OX₂ Receptor OX₁ Receptor

Actividad biológica
Pureza y Documentación
Referencias
Revisión del cliente

Descripciòn	Cleminorexton is an orally active orexin-2 receptor (OX2R) agonist with a pEC₅₀ between 9 and 10.4. Cleminorexton can be used for narcolepsy and other conditions associated with orexin deficiency and/or excessive sleepiness^[1].
In Vivo	Cleminorexton (Compound 67A/Example 47) (1-10 mg/kg, p.o., single dose) shows significant arousal-promoting activity in mouse models^[1]. MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Peso molecular	512.52
Fòrmula	C₂₄H₂₄F₄N₂O₄S
No. CAS	2980518-93-0
SMILES	FC1=C(C2=C(C(F)=CC(F)=C2)OCCC3=O)C=CC=C1C[C@]4([H])N3CCC[C@@]4(NS(C5(CC5)F)(=O)=O)[H]
Envío	Room temperature in continental US; may vary elsewhere.
Almacenamiento	Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación	Ficha de datos (269 KB) SDS (252 KB) Instrucciones de manejo (2659 KB)
Referencias	[1]. Gregory R. Ott, et al., Medium- or macro-cyclic benzyl-substituted heterocycle derivatives and related uses. WO2023167925A1.

Cleminorexton Related Classifications

Neurological Disease Metabolic Disease

Calculadora de molaridad
Calculadora de dilución

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass		Concentration		Volume		Molecular Weight *
	=		×		×

The dilution calculator equation

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Cleminorexton2980518-93-0Orexin Receptor (OX Receptor)Hypocretin ReceptorHCRT ReceptorInhibitorinhibitorinhibit

Productos vistos recientemente:

Nombre del producto

Requested Quantity *

Nombre del solicitante *

Saludo

Direcciòn del E-mail *

Número de teléfono *

Department

Nombre de la Organizaciòn *

City

Provincia

Country or Region *

Observaciones

Nombre del producto

Lot #

Nombre del solicitante *

Direcciòn del E-mail *

Número de teléfono

Department *

Nombre de la Organizaciòn *

Country or Region *

Observaciones

Name
E-mail *

	Sorry, but the email address you supplied was invalid.

Cleminorexton

Cleminorexton Related Antibodies

Recomendaciones destacadas

•Related Small Molecules:

•Related Proteins:

Ver todos los productos específicos de isoformas Orexin Receptor (OX Receptor):

Actividad biológica

Pureza y Documentación

Referencias

Revisión del cliente

Cleminorexton Related Classifications

Calculadora de molaridad

Calculadora de dilución