2. GPCR/G Protein
  3. GHSR
  4. Ghrelin receptor full agonist-2

Ghrelin receptor full agonist-2 (compound 12j) is a highly potent Ghrelin receptor full agonist.

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Ghrelin receptor full agonist-2

Ghrelin receptor full agonist-2 Chemische Struktur

CAS. Nr. : 2602452-73-1

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Ghrelin receptor full agonist-2 Related Antibodies

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Beschreibung

Ghrelin receptor full agonist-2 (compound 12j) is a highly potent Ghrelin receptor full agonist.

Cellular Effect
Cell Line Type Value Description References
HEK293 EC50
0.442 1
Compound: 12j
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
HEK293 EC50
0.442 1
Compound: 12j
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
HEK293 EC50
0.442 1
Compound: 12j
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
HEK293 EC50
0.9 1
Compound: 12j
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
HEK293 EC50
0.9 1
Compound: 12j
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
HEK293 EC50
0.9 1
Compound: 12j
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
Molekulargewicht

558.05

Formel

C26H28ClN5O5S
CAS. Nr.
SMILES

O=C(C1=NOC(C2=C(C=CC=C2)Cl)=C1)N[C@@H]3[C@H](CN(C3)S(=O)(C4=CC=CC=C4)=O)C(N[C@H]5CCCNC5)=O
Versand

Room temperature in continental US; may vary elsewhere.
Speicherung

Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
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Ghrelin receptor full agonist-2 Related Classifications

  • Molaritätsrechner

  • Verdünnungsrechner

Die Formel zur Berechnung von Molaritäten

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)

Diese Gleichung wird häufig abgekürzt als: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Ghrelin receptor full agonist-22602452-73-1Ghrelin receptor full agonist2Ghrelin receptor full agonist 2GHSRGrowth hormone secretagogue receptorGhrelin receptorInhibitorinhibitorinhibit

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