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Results for "

A1AR Agonist

" in MedChemExpress (MCE) Product Catalog:
Cat. No. 상품명 Target 연구분야 Chemical Structure
  • HY-103180
    2'-MeCCPA

    2-Chloro-N-cyclopentyl-2′-C-methyladenosine

    		 Adenosine Receptor Neurological Disease
    2'-MeCCPA is a potent and selective A1 adenosine receptors (A1AR) agonist. 2'-MeCCPA efficiently inhibits cAMP modulation in both direct pathway medium spiny neurons (dMSNs) and indirect pathway medium spiny neurons (iMSNs) .
    2'-MeCCPA
  • HY-101854
    N6-(2-Phenylethyl)adenosine

    N6-Phenethyladenosine; N6-Phenylethyladenosine

    		 Adenosine Receptor Inflammation/Immunology Cancer
    N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine), an adenosine derivative, is a potent adenosine receptors (AR) agonist with Ki values of 11.8 nM, 30.1 nM, 0.63 nM for rat A1AR, human A1AR and hA3AR, respectively .
    N6-(2-Phenylethyl)adenosine
  • HY-112567
    TRR469

    		Adenosine Receptor Neurological Disease
    TRR469 is a positive allosteric modulator of the A1 adenosine receptor (A1AR). TRR469 significantly increases the affinity of 2-chloro N(6)-cyclopentyladenosine (CCPA) for A₁AR, increasing the number of receptors recognized by the agonist radioligand [³H]-CCPA. TRR469 shows significant effects in both anxiety and pain models. TRR469 can be used to study anxiety disorders and pain management .
    TRR469
  • HY-103163
    (±)-5'-Chloro-5'-deoxy-ENBA

    		Adenosine Receptor Neurological Disease
    (±)-5'-Chloro-5'-deoxy-ENBA is an agonist of A1AR. (±)-5'-Chloro-5'-deoxy-ENBA produces hypothermia in mice .
    (±)-5'-Chloro-5'-deoxy-ENBA
  • HY-106186
    GW-493838

    		Adenosine Receptor Neurological Disease
    GW-493838 is a potent Adenosine A1 (A1AR) agonist. GW-493838 has the potential for the research of neuropathic pain .
    GW-493838
  • HY-182687
    MRS7469

    		Adenosine Receptor Neurological Disease
    MRS7469 is a highly selective A1 adenosine receptor (A1AR) agonist with over 2000-fold selectivity over other adenosine receptor subtypes. MRS7469 stably binds to the orthosteric binding site of A1AR, and exhibits extremely high affinity for both humans and mice (e.g., human pKi is 8.67, mouse pKi is 9.43). By activating central A1AR, MRS7469 significantly induces hypothermia, motor inhibition and psychomotor dysfunction, and can be widely used in research related to depression and other relevant fields .
    MRS7469
  • HY-101854R
    N6-(2-Phenylethyl)adenosine (Standard)

    N6-Phenethyladenosine (Standard); N6-Phenylethyladenosine (Standard)

    		 Reference Standards Adenosine Receptor Inflammation/Immunology Cancer
    N6-(2-Phenylethyl)adenosine (Standard) (N6-Phenethyladenosine (Standard)) is the analytical standard of N6-(2-Phenylethyl)adenosine (HY-101854). This product is intended for research and analytical applications. N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine), an adenosine derivative, is a potent adenosine receptors (AR) agonist with Ki values of 11.8 nM, 30.1 nM, 0.63 nM for rat A1AR, human A1AR and hA3AR, respectively .
    N6-(2-Phenylethyl)adenosine (Standard)
  • HY-W069173
    2-Thioadenosine

    		Adenosine Receptor Others
    2-Thioadenosine is a selective A1 adenosine receptor (A1AR) ligand with a Ki of 80.3 nM. 2-Thioadenosine shows very low affinity for the A2A, A2B and A3 adenosine receptor subtypes. 2-Thioadenosine acts as a precursor for the synthesis of fluorescent A3 adenosine receptor-selective agonists .
    2-Thioadenosine

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