2. Metabolic Enzyme/Protease
  3. Isocitrate Dehydrogenase (IDH)
  4. Mutant IDH1-IN-4

Mutant IDH1-IN-4 (compound 434) is an inhibitor of mutant Isocitrate dehydrogenase 1 (IDH 1), with IC50 values of ≤ 0.5 μM for mutant IDH1 in R132H, HT1080 and U87R132H cells.

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Mutant IDH1-IN-4

Mutant IDH1-IN-4 화학구조

CAS No. : 1416270-18-2

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10 mg   견적 받기  
50 mg   견적 받기  

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Mutant IDH1-IN-4 Related Antibodies

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제품 설명

Mutant IDH1-IN-4 (compound 434) is an inhibitor of mutant Isocitrate dehydrogenase 1 (IDH 1), with IC50 values of ≤ 0.5 μM for mutant IDH1 in R132H, HT1080 and U87R132H cells[1].

IC50 & Target

IC50: ≤ 0.5 μM (mutant IDH 1 in cells)[1].
분자량

438.56

화학식

C25H34N4O3
CAS No.
Appearance

Solid

Color

Light yellow to yellow

SMILES

N#CC1=C(N2C[C@@H](C3CC3)N(C(CCOC)=O)CC2)N=C(C4CC4)C5=C1CC(C)(C)OC5
선적

Room temperature in continental US; may vary elsewhere.
보관
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
순도&문서
References
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Mutant IDH1-IN-4 Related Classifications

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The molarity calculator equation

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Mutant IDH1-IN-41416270-18-2Isocitrate Dehydrogenase (IDH)Inhibitorinhibitorinhibit

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상품명:
Mutant IDH1-IN-4
Cat. No.:
HY-114459
수량:
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SAFETY DATA SHEET (SDS)

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