1. GPCR/G Protein
  2. Oxytocin Receptor

PF-3274167 (Synonyms: cligosiban)

Cat. No.: HY-15023 Purity: 99.40%
Handling Instructions

PF-3274167 is a high-affinity nonpeptide oxytocin receptor (OTR) antagonist, with Ki of 9.5 nM.

For research use only. We do not sell to patients.

PF-3274167 Chemical Structure

PF-3274167 Chemical Structure

CAS No. : 900510-03-4

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 238 In-stock
Estimated Time of Arrival: December 31
5 mg USD 216 In-stock
Estimated Time of Arrival: December 31
10 mg USD 312 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1152 In-stock
Estimated Time of Arrival: December 31
100 mg USD 1920 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

PF-3274167 is a high-affinity nonpeptide oxytocin receptor (OTR) antagonist, with Ki of 9.5 nM. IC50 value: 9.5 nM [1] Target: oxytocin receptor (OTR)

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.3819 mL 11.9093 mL 23.8186 mL
5 mM 0.4764 mL 2.3819 mL 4.7637 mL
10 mM 0.2382 mL 1.1909 mL 2.3819 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

419.84

Formula

C₁₉H₁₉ClFN₅O₃

CAS No.

900510-03-4

SMILES

FC1=CC(Cl)=C(OC2CN(C3=NN=C(COC)N3C4=CC=C(OC)N=C4)C2)C=C1

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Inquiry Information

Product Name:
PF-3274167
Cat. No.:
HY-15023
Quantity:

PF-3274167

Cat. No.: HY-15023