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Drug Derivative

Drug derivative

Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.

Drug Derivative Produits associés (3817):

Cat. No. Nom du produit Effet Pureté Chemical Structure
  • HY-139420R
    Tafluprost ethyl amide (Standard)
    Tafluprost ethyl amide (Standard) is the analytical standard of Tafluprost ethyl amide (HY-139420). This product is intended for research and analytical applications. Tafluprost ethyl amide is a derivative of Tafluprost (HY-B0600). Tafluprost ethyl amide is commonly used in studies related to eyelash hypotrichosis, and it can also be applied in research related to the cosmetic field.
    Tafluprost ethyl amide (Standard)
  • HY-W975617
    4',5,7,8-Tetrahydroxyflavanone
    4',5,7,8-Tetrahydroxyflavanone is an isocarthamidin compound.
    4',5,7,8-Tetrahydroxyflavanone
  • HY-W715341R
    RO-1-5237 (Standard)
    RO-1-5237 (Standard) is the analytical standard of RO-1-5237. This product is intended for research and analytical applications. RO-1-5237 is a metabolite of Pyridostigmine Bromide, which is a cholinergic and can be used for myasthenia gravis research.
    RO-1-5237 (Standard)
  • HY-133597R
    4-Chlorocatechol (Standard)
    4-Chlorocatechol (Standard) is the analytical standard of 4-Chlorocatechol. This product is intended for research and analytical applications. 4-Chlorocatechol is a major degradation product of 4-chloro-2-aminophenol (4C2AP). 4-Chlorocatechol is also a substrate for catechol 1,2-dioxygenases and chlorocatechol dioxygenase.
    4-Chlorocatechol (Standard)
  • HY-N18876
    Homostephanoline
    Homostephanoline is a corydane-type alkaloid that can be isolated from species of the Stephania subgenus.
    Homostephanoline
  • HY-172074
    N-Propylnorketamine hydrochloride
    N-Propylnorketamine hydrochloride is structurally categorized as an arylcyclohexylamine.
    N-Propylnorketamine hydrochloride
  • HY-W701712
    Fenamiphos sulfone
    Fenamiphos sulfone is the oxidative metabolite of the organophosphorus pesticide fenamiphos. Fenamiphos sulfone undergoes biotransformation and accumulates in aquatic and terrestrial algal species.
    Fenamiphos sulfone
  • HY-129881
    2-Thiothinone hydrochloride
    2-Thiothinone hydrochloride is a thiophene.
    2-Thiothinone hydrochloride
  • HY-163836
    HMBPP analog 1
    HMBPP analog 1 (6e), a Trifluoromethyl analog, is the weakest agonist but the strongest inhibitor HMBPP ELISA response.
    HMBPP analog 1
  • HY-132002
    Dimethylsildenafil
    Dimethylsildenafil is a derivative of Sildenafil (HY-15025). Sildenafil is a potent phosphodiesterase type 5 (PDE5) inhibitor with an IC50 of 5.22 nM.
    Dimethylsildenafil
  • HY-172002
    3'-O-Methylguanosine-5'-O-triphosphate sodium
    3'-O-Methylguanosine-5'-O-triphosphate (3'-O-Methyl GTP) sodium is a methylated derivative of Guanosine 5'-triphosphate (HY-W010737). 3'-O-Methylguanosine-5'-O-triphosphate has been used as a chain termination reagent in the preparation of early RNA polymerase II elongation intermediates.
    3'-O-Methylguanosine-5'-O-triphosphate sodium
  • HY-168759
    11α-Hydroxytestosterone
    11α-Hydroxytestosterone is a deriviative of Hydrocortisone (HY-N0583), with the relative binding affinity to progesterone receptor of 9% (comparing to R5020 (HY-119384) 100%). 11α-Hydroxytestosterone inhibits the growth and differentiation of human decidual cells in culture.
    11α-Hydroxytestosterone
  • HY-N19809
    10-Deacetyl-10-oxo-7-epi-taxol
    10-Deacetyl-10-oxo-7-epi-taxol is a cytotoxic agent with a 9,10-diketone structure. 10-Deacetyl-10-oxo-7-epi-taxol induces cytotoxic activity in cancer cells.
    10-Deacetyl-10-oxo-7-epi-taxol
  • HY-183865
    F1414-1444
    F1414-1444 is a DBPI skeleton derivative and a potent inhibitor of IspQ (Rv0338c)-targeting Mycobacterium tuberculosis. F1414-1444 binds to the membrane-bound iron-sulfur oxidoreductase IspQ, induces oxidative stress and thiol stress in bacterial cells, upregulates the expression of stress-related genes such as the SigK regulon, thereby inhibiting bacterial proliferation and exerting bactericidal activity. F1414-1444 only inhibits the Mycobacterium tuberculosis complex and Mycobacterium marinum. F1414-1444 can be used in studies related to Mycobacterium tuberculosis.
    F1414-1444
  • HY-W709830
    α-Propylaminopentiophenone hydrochloride
    		Control
    α-Propylaminopentiophenone hydrochloride is a drug derivative.
    α-Propylaminopentiophenone hydrochloride
  • HY-W701713
    Fenamiphos sulfoxide
    Fenamiphos sulfoxide is the major oxidative metabolite of the organophosphate pesticide fenamiphos. Fenamiphos sulfoxide can be transformed by aquatic and terrestrial algae, and undergoes bioaccumulation in these organisms.
    Fenamiphos sulfoxide
  • HY-172077
    4-MA-NBOMe hydrochloride
    4-MA-NBOMe hydrochloride is structurally categorized as an amphetamine.
    4-MA-NBOMe hydrochloride
  • HY-172001
    α-GalCer analog 8
    α-GalCer analog 8 is a triazole derivative of α-Galactosylceramide (HY-102022). α-Galactosylceramide is a synthetic glycolipid with antitumorial and immunostimulatory.
    α-GalCer analog 8
  • HY-117109R
    Amino Tadalafil (Standard)
    Amino Tadalafil (Standard) is the analytical standard of Amino Tadalafil. This product is intended for research and analytical applications. Amino Tadalafil is a structural analogue of Tadalafil (HY-90009A). Tadalafil is a potent inhibitor of PDE5 with applications in several conditions, including erectile dysfunction, pulmonary arterial hypertension, and lower urinary tract dysfunction.
    Amino Tadalafil (Standard)
  • HY-115231
    ci-IP3/PM
    ci-IP3/PM is a caged and cell permeable derivative of IP3. ci-IP3/PM can induce Ca2+ release from internal stores.
    ci-IP3/PM