2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. Herkinorin

Herkinorin is a potent and selective agonist of µ opioid receptor with a Ki of 45 nM Herkinorin is widely used for pain research.

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Herkinorin

Herkinorin Estructura química

No. CAS : 862073-77-6

Tamaño Precio Stock Cantidad
500 μg Obtener un presupuesto 3 - 4 Weeks 4 - 5 Weeks 5 - 6 Weeks 2 - 3 weeks
1 mg Obtener un presupuesto 3 - 4 Weeks 4 - 5 Weeks 5 - 6 Weeks 2 - 3 weeks
5 mg   Obtener un presupuesto  
10 mg   Obtener un presupuesto  
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Based on 1 publication(s) in Google Scholar

Herkinorin Related Antibodies

Top Publications Citing Use of Products

1 Publications Citing Use of MCE Herkinorin

Ver todos los productos específicos de isoformas Opioid Receptor:

Ver todas las isoformas
μ Opioid Receptor/MOR κ Opioid Receptor/KOR δ Opioid Receptor/DOR NOP Receptor/ORL1

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Descripciòn

Herkinorin is a potent and selective agonist of µ opioid receptor with a Ki of 45 nM Herkinorin is widely used for pain research[1].

Cellular Effect
Cell Line Type Value Description References
CHO EC50
1320 nM
Compound: 1c
Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
[PMID: 18380425]
CHO EC50
1320 nM
Compound: 13
Stimulation of [35S]GTP-gamma-S, binding to Opioid receptor kappa1 expressed in CHO cells
Stimulation of [35S]GTP-gamma-S, binding to Opioid receptor kappa1 expressed in CHO cells
[PMID: 16033256]
CHO EC50
500 nM
Compound: 1c
Agonist activity at human recombinant mu opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
Agonist activity at human recombinant mu opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
[PMID: 18380425]
CHO EC50
500 nM
Compound: 13
Stimulation of [35S]GTP-gamma-S, binding to Opioid receptor mu1 expressed in CHO cells
Stimulation of [35S]GTP-gamma-S, binding to Opioid receptor mu1 expressed in CHO cells
[PMID: 16033256]
Peso molecular

494.53

Fòrmula

C28H30O8
No. CAS
SMILES

O=C([C@H](C[C@H](OC(C1=CC=CC=C1)=O)C([C@@]23[H])=O)[C@]2(C)CC[C@@]([C@]3(C)C[C@@H](C4=COC=C4)O5)([H])C5=O)OC
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
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Herkinorin Related Classifications

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Herkinorin862073-77-6Opioid ReceptorInhibitorinhibitorinhibit

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Nombre del producto:
Herkinorin
Cat. No.:
HY-121415
Cantidad:
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