μ Opioid Receptor/MOR

μ Opioid Receptor/MOR Related Products (29):

By Type:	Pan (4) Selective (10)
By Effects:	Inhibitors (2) Agonists (14) Antagonists (10) Activator (1) Modulator (1)

Cat. No.	Product Name	Effect	Purity

HY-N0164

Matrine	Agonist	≥98.0%
Matrine (Matridin-15-one) is an alkaloid found in plants from the Sophora genus that can act as a kappa opioid receptor and u-receptor agonist.

HY-15122A

Sinomenine hydrochloride	Activator	99.88%
Sinomenine hydrochloride (Cucoline hydrochloride), an alkaloid extracted from Sinomenium acutum, is a blocker of the NF-κB activation.

HY-P0185

Endomorphin 1	Agonist	99.92%
Endomorphin 1, a high affinity, highly selective agonist of the μ-opioid receptor (K_i: 1.11 nM), displays reasonable affinities for kappa₃ binding sites, with K_i value between 20 and 30 nM.

HY-124754

Navacaprant	Inhibitor	99.71%
Navacaprant (BTRX-335140) is a selective and orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC₅₀ values of 0.8 nM, 110 nM, and 6500 nM, respectively.

HY-P1335A

CTAP TFA	Antagonist	99.56%
CTAP TFA is a potent, highly selective, and BBB penetrant μ opioid receptor antagonist, with an IC₅₀ of 3.5 nM.

HY-P0185A

Endomorphin 1 acetate	Agonist	99.92%
Endomorphin 1 acetate, a high affinity, highly selective agonist of the μ-opioid receptor (K_i: 1.11 nM), displays reasonable affinities for kappa₃ binding sites, with K_i value between 20 and 30 nM.

HY-151811

NAQ	Agonist
NAQ is a potent and selective μ opioid receptor partial agonist, with a K_i of 0.55 nM.

HY-114072

J-113397	Antagonist
J-113397 is the first potent and selective nonpeptidyl ORL1 receptor antagonist (K_i: cloned human ORL1=1.8 nM) without any agonistic effects on other opioid receptors.

HY-P0244

Dermorphin	Agonist	98.06%
Dermorphin is a natural heptapeptide μ-opioid receptor (MOR) agonist found in amphibian skin.

HY-N0923

Corydaline	Agonist	98.44%
Corydaline ((+)-Corydaline), an isoquinoline alkaloid isolated from Corydalis yanhusuo, is an AChE inhibitor with an IC₅₀ of 226 µM.

HY-P1329A

CTOP TFA	Antagonist	99.93%
CTOP TFA is a potent and highly selective μ-opioid receptor antagonist.

HY-P1087

Adrenorphin	Agonist
Adrenorphin is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with K_i of 12 nM.

HY-P1866A

β-Endorphin, equine TFA	Agonist
β-Endorphin, equine TFA is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors.

HY-P1701

Morphiceptin		99.35%
Morphiceptin is a potent and specific agonist for morphine (μ) receptors.

HY-107748

5'-Guanidinonaltrindole hydrochloride	Antagonist	98.65%
5'-Guanidinonaltrindole (5'-GNTI) hydrochloride is a highly selective and potent κ-opioid receptor antagonist with a K_i of 0.18 nM for human κ-opioid receptor.

HY-N0398

Sec-O-Glucosylhamaudol	Inhibitor	99.89%
Sec-O-Glucosylhamaudol is a natural compound extracted from Peucedanum japonicum Thunb, decreases levels of μ-opioid receptor, with analgesic effect.

HY-101011

Naloxonazine dihydrochloride	Antagonist
Naloxonazine dihydrochloride is a specific μ-opioid receptor antagonist with an IC₅₀ of 5.4 nM.

HY-141515

BMS-986121	Modulator	98.89%
BMS-986121 is a positive allosteric modulator (PAM) of the μ opioid receptor extracted from patent WO2014107344.

HY-115066

GSK1521498 free base	Antagonist	98.55%
GSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist.

HY-P1335

CTAP	Antagonist
CTAP is a potent, highly selective, and BBB penetrant μ opioid receptor antagonist, with an IC₅₀ of 3.5 nM.

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