2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. UCM707

UCM707, a potent and selective inhibitor of endocannabinoid uptake, potentiates hypokinetic and antinociceptive effects of Anandamide.

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UCM707

UCM707 Chemical Structure

CAS No. : 390824-20-1

Size Prix Stock Quantité
1 mg Obtenir un devis 2 - 3 weeks 4 - 5 weeks 5 - 6 weeks 1 - 2 weeks
5 mg Obtenir un devis 2 - 3 weeks 4 - 5 weeks 5 - 6 weeks 1 - 2 weeks
10 mg Obtenir un devis 2 - 3 weeks 4 - 5 weeks 5 - 6 weeks 1 - 2 weeks
50 mg   Obtenir un devis  
100 mg   Obtenir un devis  
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UCM707 Related Antibodies

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Description

UCM707, a potent and selective inhibitor of endocannabinoid uptake, potentiates hypokinetic and antinociceptive effects of Anandamide[1].

Cellular Effect
Cell Line Type Value Description References
U-937 IC50
0.8 μM
Compound: 42
Concentration required to inhibit anandamide uptake in U937 cell line
Concentration required to inhibit anandamide uptake in U937 cell line
[PMID: 16078824]
U-937 IC50
0.8 μM
Compound: 5
Inhibition of [3H]anandamide transport(ANT) in human lymphoma U937 cell
Inhibition of [3H]anandamide transport(ANT) in human lymphoma U937 cell
[PMID: 12672252]
U-937 IC50
0.8 μM
Compound: 9
Ability to inhibit [3H]anandamide uptake in human lymphoma U937 cells
Ability to inhibit [3H]anandamide uptake in human lymphoma U937 cells
[PMID: 11741470]
U-937 IC50
1.46 μM
Compound: UCM707
Inhibition of [ethanol-amine-1-3H]AEA uptake in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liquid scintillation counting
Inhibition of [ethanol-amine-1-3H]AEA uptake in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liquid scintillation counting
[PMID: 24972328]
U-937 IC50
7.24 μM
Compound: UCM707
Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liquid scintillation counting
Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liquid scintillation counting
[PMID: 24972328]
Masse moléculaire

383.57

Formule

C25H37NO2
CAS No.
SMILES

CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(NCC1=COC=C1)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
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UCM707 Related Classifications

  • Calculateur de molarité

  • Calculateur de dilution

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

UCM707390824-20-1UCM 707UCM-707Cannabinoid Receptorendocannabinoid uptakehypokineticantinociceptive effectInhibitorinhibitorinhibit

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