CB1

CB1 Related Products (55):

By Type:	Pan (14) Selective (31)
By Effects:	Inhibitors (8) Agonists (24) Antagonists (16) Activator (1) Modulators (5)

Cat. No.	Product Name	Effect	Purity

HY-14137

Rimonabant Hydrochloride	Antagonist	99.95%
Rimonabant Hydrochloride (SR 141716A Hydrochloride) is a highly potent and selective central cannabinoid receptor (CB1) antagonist with an K_i of 1.8 nM.

HY-18697

JD-5037	Antagonist	98.05%
JD-5037 is a potent CB₁R antagonist with an IC₅₀ of 1.5 nM.

HY-B0151

Pregnenolone	Inhibitor	98.05%
Pregnenolone (3β-Hydroxy-5-pregnen-20-one) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones.

HY-112340

TM38837	Antagonist	99.00%
TM38837 is a peripheral selective cannabinoid receptor type 1 (CB1) receptor antagonist.

HY-110189

Pregnenolone monosulfate sodium	Inhibitor
Pregnenolone monosulfate sodium (3β-Hydroxy-5-pregnen-20-one monosulfate sodium) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones.

HY-P99755

Nimacimab	Inhibitor
Nimacimab (RYI-018) is a negative-allosteric modulating monoclonal antibody targeting CB1 receptor.

HY-148176

ANEB-001	Inhibitor
ANEB-001 is an orally active CB1 inhibitor, can be used to research acute cannabinoid intoxication.

HY-152254

CB2R/FAAH modulator-3	Agonist	99.71%
CB2R/FAAH modulator-3 (compound 27) is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor.

HY-100488

Bay 59-3074	Agonist	99.00%
Bay 59-3074 is a selective cannabinoid CB₁/CB₂ receptor partial agonist with K_i values of 48.3 and 45.5 nM at human CB₁ and CB₂ receptors, respectively.

HY-13505

AM281	Antagonist	≥99.0%
AM281 is a selective CB1 receptor antagonist with an IC₅₀ of 9.91 nM.

HY-W005629

Leelamine	Agonist	98.36%
Leelamine is a weak agonist of cannabinoid receptors CB1 and CB2.

HY-113204

N-Oleoyl glycine	Activator	≥99.0%
N-Oleoyl glycine is a lipoamino acid, which stimulates adipogenesis associated with activation of CB1 receptor and Akt signaling pathway in 3T3-L1 adipocyte.

HY-B1739

Pregnenolone monosulfate	Inhibitor	≥98.0%
Pregnenolone monosulfate (3β-Hydroxy-5-pregnen-20-one monosulfate) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones.

HY-N0919

Yangonin	Inhibitor	99.79%
Yangonin exhibits affinity for the human recombinant cannabinoid CB1 receptor with an IC₅₀ and a K_i of 1.79 μM and 0.72 μM, respectively.

HY-119104

AZD1940	Agonist	99.45%
AZD1940 is an orally active, high affinity cannabinoid CB1/CB2 receptor agonist with pK_i values of 7.93 and 9.06 for human CB1R and CB2R, respectively.

HY-110028

Leelamine hydrochloride	Agonist	98.10%
Leelamine hydrochloride is a tricyclic diterpene molecule that is extracted from the bark of pine trees.

HY-P1397A

RVD-Hpα TFA	Agonist	98.99%
RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.

HY-113689

GAT211	Agonist	99.98%
GAT211 is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM).

HY-116637

Tetrahydromagnolol	Agonist	99.79%
Tetrahydromagnolol (Magnolignan), a main metabolite of Magnolol, is a potent and selective cannabinoid CB2 receptor agonist with an EC₅₀ of 170 nM and a K_i of 416 nM.

HY-14136

Rimonabant	Antagonist
Rimonabant (SR141716) is a highly potent, brain penetrated and selective central cannabinoid receptor (CB1) antagonist with a K_i of 1.8 nM.

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