CB1 Agonist

CB1 Agonists (24):

Cat. No.	Product Name	Effect	Purity

HY-152254

CB2R/FAAH modulator-3	Agonist	99.71%
CB2R/FAAH modulator-3 (compound 27) is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor.

HY-152253

CB2R/FAAH modulator-2	Agonist
CB2R/FAAH modulator-2 (compound 26) is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor.

HY-100488

Bay 59-3074	Agonist	99.00%
Bay 59-3074 is a selective cannabinoid CB₁/CB₂ receptor partial agonist with K_i values of 48.3 and 45.5 nM at human CB₁ and CB₂ receptors, respectively.

HY-110028

Leelamine hydrochloride	Agonist	98.10%
Leelamine hydrochloride is a tricyclic diterpene molecule that is extracted from the bark of pine trees.

HY-W005629

Leelamine	Agonist	98.36%
Leelamine is a weak agonist of cannabinoid receptors CB1 and CB2.

HY-P1397A

RVD-Hpα TFA	Agonist	98.99%
RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.

HY-113689

GAT211	Agonist	99.98%
GAT211 is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM).

HY-110014

Noladin ether	Agonist	≥98.0%
Noladin ether is a potent and selective agonist of cannabinoid CB₁ receptor, with a K_i of 21.2 nM.

HY-150029

CB1/2 agonist 3	Agonist
CB1/2 agonist 3 (compound 52), a potent non-selective cannabinoid ligand, is a CB1/CB2 (cannabinoid receptor) competitive agonist.

HY-110036

GW-405833	Agonist	99.12%
GW-405833 (L768242) is a potent, selective cannabinoid receptor 2 (CB₂) agonist with an EC₅₀ of 50.7 nM.

HY-116637

Tetrahydromagnolol	Agonist	99.79%
Tetrahydromagnolol (Magnolignan), a main metabolite of Magnolol, is a potent and selective cannabinoid CB2 receptor agonist with an EC₅₀ of 170 nM and a K_i of 416 nM.

HY-119104

AZD1940	Agonist	99.45%
AZD1940 is an orally active, high affinity cannabinoid CB1/CB2 receptor agonist with pK_i values of 7.93 and 9.06 for human CB1R and CB2R, respectively.

HY-147512

CB1/2 agonist 1	Agonist
CB1/2 agonist 1 is a potent and cross the blood-brain barrier CB1/2 agonist with EC₅₀s of 56.15, 11.63 nM for CB1R and CB2R, respectively.

HY-112707

AM9405	Agonist
AM9405 is a novel peripherally active cannabinoid type 1 (CB1) and serotonin type 3 receptor agonist.

HY-119744

BAY 38-7271	Agonist
BAY 38-7271 is selective and highly potent and cannabinoid CB₁/CB₂ receptor agonist, with K_is of 1.85 nM and 5.96 nM for recombinant human CB₁ receptor and CB₂ receptor, respectively.

HY-151107

CBR Agonist-2	Agonist
CBR Agonist-2 is a CB1 agonist (CB1R; CB1 ligand) with an EC₅₀ and a K_i of 960 nM and 970 nM, respectively.

HY-150067

CB1R antagonist 1	Agonist
CB1R Allosteric modulator 5, a selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC₅₀ value of 4.2 μM and EC₅₀ value of ＞10 μM.

HY-12095

CB1 inverse agonist 2	Agonist
CB1 inverse agonist 2 is an orally active inverse agonist of Cannabinoid Receptor CB1.

HY-W013788

2-Palmitoylglycerol	Agonist	≥99.0%
2-Palmitoylglycerol (2-Palm-Gl), an congener of 2-arachidonoylglycerol (2-AG), is a modest cannabinoid receptor CB1 agonist.

HY-152251

CB2R/FAAH modulator-1	Agonist
CB2R/FAAH modulator-1 is a cannabinoid type 2 receptor (CB2R) full agonist with K_is of 14.8 nM and 241.3 nM for CB2R and CB1R, respectively.

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