1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Cannabinoid Receptor
  4. CB2 Inhibitors

CB2 Inhibitors

CB1

CB2

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform CB2 together.

Please try each isoform separately.

CB2 Specific Inhibitors, Agonists, Antagonists & Modulators
Product Name CB2 CB1 CB2 Selectivity Purity
Bay 59-3074
CB2 , Ki: 45.5 nM
CB1 , Ki: 48.3 nM
Selective Agonist 98.85%
CB2R-IN-1
CB2 , Ki: 0.9 nM
  Selective Inhibitor
Tedalinab
CB2
  Selective Inhibitor
Ibipinabant
CB2 , Ki: 7943 nM
CB1 , Ki: 7.8 nM
Selective Antagonist
PM226
CB2 , EC50: 39 nM
CB2 , Ki: 13 nM
  Selective Agonist
Tetrahydromagnolol
CB2 , EC50: 170 nM
CB2 , Ki: 416 nM
CB1 , EC50: 9010 nM
CB1 , Ki: 2260 nM
Selective Agonist
AZD1940
hCB2-R, pKi: 9.06
hCB1-R, pKi: 7.93
Pan Agonist 99.45%
EHP-101
CB2
  Pan Agonist 98.56%
LY320135
CB2 , Ki: >10 μM
CB1 , Ki: 141 nM
Pan Antagonist
AM281
CB2 , IC50: 13000 nM
CB1 , IC50: 9.91 nM
Pan Antagonist
Drinabant
CB2 , IC50: 10000 nM
rCB1-R, IC50: 10 nM
hCB1-R, IC50: 25 nM
Pan Antagonist
BAY 38-7271
CB2 , Ki: 5.96 nM
CB1 , Ki: 1.85 nM
Pan Agonist
CB2 modulator 1
CB2
  Modulator
CB2R PAM
cannabinoid type-2 receptors
  Agonist