1. GPCR/G Protein
  2. Cholecystokinin Receptor

CHEMBL333994 (Synonyms: FK-480)

Cat. No.: HY-U00363
Handling Instructions

CHEMBL333994 is a potent and orally effective Cholecystokinin A (CCK-A) antagonist, with an IC50 of 0.67 nM.

For research use only. We do not sell to patients.

CHEMBL333994 Chemical Structure

CHEMBL333994 Chemical Structure

CAS No. : 167820-10-2

Size Price Stock
1 mg USD 1536 Get quote
5 mg USD 3072 Get quote
10 mg USD 5220 Get quote
20 mg USD 9216 Get quote

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

CHEMBL333994 is a potent and orally effective Cholecystokinin A (CCK-A) antagonist, with an IC50 of 0.67 nM.

IC50 & Target

IC50: 0.67 nM(CCK-A)[1].

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2808 mL 11.4038 mL 22.8076 mL
5 mM 0.4562 mL 2.2808 mL 4.5615 mL
10 mM 0.2281 mL 1.1404 mL 2.2808 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

438.45

Formula

C₂₆H₁₉FN₄O₂

CAS No.

167820-10-2

SMILES

O=C(C(N1)=CC2=C1C=CC=C2)N[[email protected]]3C(N4C5=C(CC4)C=CC=C5C(C6=CC=CC=C6F)=N3)=O

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
CHEMBL333994
Cat. No.:
HY-U00363
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CHEMBL333994

Cat. No.: HY-U00363