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Cat. No.: HY-U00363A

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(rac)-CHEMBL333994

(Synonyms: (rac)-FK-480)

(rac)-CHEMBL333994 is the racemate of CHEMBL333994 (HY-U00363). CHEMBL333994 is a potent and orally active Cholecystokinin A receptor (CCK-A receptor) antagonist, with an IC₅₀ of 0.67 nM. CHEMBL333994 selectively antagonizes peripheral CCK receptors. CHEMBL333994 increases CCK mRNA level. CHEMBL333994 can be used for research of chronic pancreatitis.

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CAS No.: 126149-42-6
Formule: C₂₆H₁₉FN₄O₂
Masse moléculaire:438.45

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Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (273 KB)

(rac)-CHEMBL333994 Chemical Structure

CAS No.: 126149-42-6

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Activité biologique

Description

Voir tous les produits spécifiques à Isoform Cholecystokinin Receptor :

CCKAR
CCKBR

Chemical Information

CAS No. 126149-42-6
Masse moléculaire 438.45
Formule C₂₆H₁₉FN₄O₂
SMILES

O=C(C(N1)=CC2=C1C=CC=C2)NC3C(N4C5=C(CC4)C=CC=C5C(C6=CC=CC=C6F)=N3)=O
Synonyms

(rac)-FK-480
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

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Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (273 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Satoh Y, et al. Studies on a novel, potent and orally effective cholecystokinin A antagonist, FK-480. Synthesis and structure-activity relationships of FK-480 and related compounds. Chem Pharm Bull (Tokyo). 1994 Oct;42(10):2071-83. [Content Brief]

[2]. Funakoshi A,et al. Effect of a new cholecystokinin antagonist (FK 480) on gene expression of cholecystokinin and secretin in rat intestine. J Gastroenterol. 1994 Jun;29(3):385-7. [Content Brief]

[3]. Moriyoshi Y, et al. Duration of anti-cholecystokinin (CCK) action on the rat exocrine pancreas of new CCK receptor antagonist FK480 administered orally. J Gastroenterol. 1996 Apr;31(2):249-53 [Content Brief]

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Chemical Information
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(rac)-CHEMBL333994

Voir tous les produits spécifiques à Isoform Cholecystokinin Receptor