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ML-290 

Cat. No.: HY-112606 Purity: >98.0%
Handling Instructions

ML-290 is a first-in-class and potent relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes, with an EC50 of 94 nM.

For research use only. We do not sell to patients.

ML-290 Chemical Structure

ML-290 Chemical Structure

CAS No. : 1482500-76-4

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Description

ML-290 is a first-in-class and potent relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes, with an EC50 of 94 nM[1].

IC50 & Target

EC50: 94 nM (RXFP1)[1]

In Vitro

ML-290 is a first-in-class and potent relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes, with an EC50 of 94 nM[1].
ML290 (5 μM) shows anti-fibrotic, relaxin-like gene expression at 24 and 72 h in activated human hepatic stellate cells[1].

Molecular Weight

506.49

Formula

C₂₄H₂₁F₃N₂O₅S

CAS No.

1482500-76-4

SMILES

O=C(NC1=CC(S(=O)(C(F)(F)F)=O)=CC=C1)C2=C(NC(C3=CC=CC=C3OC(C)C)=O)C=CC=C2

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References

Purity: >98.0%

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ML-290
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HY-112606
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