1482500-76-4
1482500-76-4
Chemical Structure
ML-290
- CAS No.: 1482500-76-4
- Formula:C24H21F3N2O5S
- Molecular Weight:506.49
IUPAC Name: 2-isopropoxy-N-(2-((3-((trifluoromethyl)sulfonyl)phenyl)carbamoyl)phenyl)benzamide
InChIKey: RSYHJSDOGMSLDH-UHFFFAOYSA-N
SMILES: O=C(NC1=CC(S(=O)(C(F)(F)F)=O)=CC=C1)C2=C(NC(C3=CC=CC=C3OC(C)C)=O)C=CC=C2
Biological Activity: ML-290 is a first-in-class and potent relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes, with an EC50 of 94 nM[1]. ML290 is a biased allosteric agonist at the relaxin receptor RXFP1.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ML-290 | 99.75% | ML-290 is a first-in-class and potent relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes, with an EC50 of 94 nM. ML290 is a biased allosteric agonist at the relaxin receptor RXFP1. | ||||||||||||||||||||
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Structural Analogs
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HY-124838EG1 -
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HY-1020673289-8625 -
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