2. Others

Others

Others

Related Products

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There are a number of inhibitors, agonists, and antagonists which we cannot make precise classification because the research area is still unknown.

Others Related Products (73787):

Cat. No. Product Name CAS No. Purity Chemical Structure
  • HY-182408
    Endosidin7 329072-88-0 98%
    Endosidin7 is a specific inhibitor for plant callose deposition during cytokinesis. Endosidin7 inhibits cytokinesis-specific callose deposition at the cell plate, disrupts cell plate maturation, and alters localization of cell plate-associated proteins during late cell plate development. Endosidin7 slows root growth and induces formation of cell wall stubs in Arabidopsis thaliana seedlings.
    Endosidin7
  • HY-182441
    (-)-AGN 192403 hydrochloride 2568912-84-3 98%
    (-)-AGN 192403 ((-)-BRD4780) hydrochloride is the enantiomer of AGN 192403 hydrochloride (HY-101374A). AGN 192403 hydrochloride is a potent and selective imidazoline-1 receptor antagonist.
    (-)-AGN 192403 hydrochloride
  • HY-182464
    DABMA 893603-33-3
    DABMA is a TMEM175 channel activator with a human EC50 of 17.9 μM. DABMA directly increases TMEM175 channel current via interaction with intracellular, transmembrane, or endosomal lumen-associated domains, and does not alter TMEM175 mRNA or protein levels. DABMA delays endolysosomal substrate degradation, modulates endolysosomal trafficking, increases acidic organelle accumulation, induces cholesterol accumulation and altered late endosome morphology. DABMA can be used for the research of coronavirus disease, Clostridium difficile infection, Pseudomonas aeruginosa infection, rabies, and influenza virus infection.
    DABMA
  • HY-182480
    Trantheline bromide 4047-34-1 98%
    Trantheline bromide is a quaternary ammonium compound. Trantheline bromide represents its intrinsic lipophilicity independent of Galvani potential difference and counter-ion effects. Trantheline bromide is used as a model compound to study the lipophilicity of quaternary ammonium ions via cyclic voltammetry.
    Trantheline bromide
  • HY-182485
    U-11634 3414-47-9 98%
    U-11634 is an orally active dopamine β-hydroxylase noncompetitive inhibitor, with rat LD50 values of 1197 mg/kg (subcutaneous) and 524 mg/kg (oral). U-11634 blocks conversion of dopamine to norepinephrine and reduces norepinephrine levels in brain. U-11634 decreases food intake and spontaneous motor activity via dietary inclusion. U-11634 induces thyroid toxicity and inhibits pregnancy. U-11634 inhibits deciduomata formation in intact and steroid-treated rats, with no reversal by progesterone or oestradiol. U-11634 can be used for pregnancy.
    U-11634
  • HY-182516
    Aminobutane bisphosphonate 32545-60-1 98%
    Aminobutane bisphosphonate is a Trypanosoma cruzi farnesyl pyrophosphate synthase (FPPS) inhibitor with an IC50 of 30.77 μM against Trypanosoma cruzi. Aminobutane bisphosphonate inhibits proliferation of intracellular amastigote Trypanosoma cruzi and lacks activity against non-infective epimastigote forms. Aminobutane bisphosphonate reduces osteoclastic bone resorption, osteoid surface extent, and osteoclast number per mm of bone surface. Aminobutane bisphosphonate can be used for the research of american trypanosomiasis (chagas' disease) and immobilization-related bone loss.
    Aminobutane bisphosphonate
  • HY-182543
    NPS-467 148717-47-9
    NPS-467 is a calcium-sensing receptor (CaR) activator and stereospecific agent with only its R-enantiomer active. NPS-467 increases the sensitivity of the CaR to activation by extracellular calcium. NPS-467 stimulates stanniocalcin (STC) secretion in trout and induces inhibition of gill calcium transport in trout. NPS-467 has no effect on serum calcitonin levels in trout.
    NPS-467
  • HY-182572
    BI 1702135 2906881-71-6 98%
    BI 1702135 is a drug intermediate that can be used to synthesize SMARCA2 PROTAC degrader BI 1810284.
    BI 1702135
  • HY-182618
    XAX-162 883053-48-3
    XAX-162 is a highly selective sphingosine 1-phosphate receptor 2 (S1PR2) agonist with a human EC50 of 0.55 μM. XAX-162 does not activate other S1P receptors. XAX-162 exhibits noncompetitive inhibition of activity by S1PR2 antagonist JTE-013 (HY-100675).
    XAX-162
  • HY-182713
    Tyrphostin AG-808 160953-95-7
    Tyrphostin AG-808 is a protein tyrosine kinase inhibitor that does not reduce neointimal formation. Perivascular implantation of Tyrphostin AG-808 causes medial damage in rats.
    Tyrphostin AG-808
  • HY-182740
    GSH linker-2
    GSH linker-2 is an ADC linker that can be used to synthesize GNE-987 GSH linker-2 (HY-138634).
    GSH linker-2
  • HY-182824
    Sucrose dilaurate 25915-57-5
    Sucrose dilaurate acts as an emulsifier, dispersant and stabilizer. Sucrose dilaurate reduces the release of HMGB1 from UVB-irradiated keratinocytes. Sucrose dilaurate inhibits melanogenesis and decreases bilirubin levels. Sucrose dilaurate induces autophagy in human epidermal keratinocytes, thereby reducing carboxymethyl lysine (CML) levels. Sucrose dilaurate reduces the secretion of insulin-like growth factor-binding protein 3 (IGFBP3) and nerve growth factor (NGF) by senescent keratinocytes. Sucrose dilaurate is investigated as an emulsifier, dispersant or stabilizer in the cosmetics, food and pharmaceutical industries.
    Sucrose dilaurate
  • HY-182934
    Cy5 MMTr CPG 1000
    Cy5 MMTr CPG 1000 is a type of fluorescently labeled solid-phase carrier used for the automated synthesis of solid-phase oligonucleotides. During the synthesis process, the Cy5 fluorescent dye can be directly covalently attached to the 3′-end of the oligonucleotide without the need for subsequent liquid-phase labeling. Cy5 MMTr CPG 1000 can be used for the synthesis of 3′-Cy5 labeled oligonucleotides.
    Cy5 MMTr CPG 1000
  • HY-182962
    7-Methylguanosine 5-disphosphoimidazolide disodium 852155-68-1 98%
    7-Methylguanosine 5-disphosphoimidazolide disodium (7-Me-3'-OMe-GDP imidazole) is a guanosine diphosphate imidazolide and starting material for synthesis of alkyne-containing C-phosphonate and phosphoester clickable mononucleotide building blocks for triazole-modified mRNA cap analogues.
    7-Methylguanosine 5-disphosphoimidazolide disodium
  • HY-182974
    DCAF1 binder 3 3033533-52-4
    DCAF1 binder 3 is a DCAF1 binder and an E3 ligase ligand. DCAF1 binder 3 can be used to synthesize PROTAC SAMHD1 Degrader-1 (HY-182970).
    DCAF1 binder 3
  • HY-182975
    E3 Ligase Ligand-linker Conjugate 229
    E3 Ligase Ligand-linker Conjugate 229 is a conjugate of an E3 ligase ligand and a linker, which can be used for the synthesis of PROTAC SAMHD1 Degrader-1 (HY-182970).
    E3 Ligase Ligand-linker Conjugate 229
  • HY-182976
    Tenovin-3-CO-C9-NH2 2917501-96-1
    Tenovin-3-CO-C9-NH2 is a conjugate of a target protein ligand and a linker, which can be used for the synthesis of PROTAC EV-A71 Degrader-1 (HY-182971).
    Tenovin-3-CO-C9-NH2
  • HY-182977
    Mal-PEG4-NPV-PABC-DMEDA
    Mal-PEG4-NPV-PABC-DMEDA is a linker that can be used for the synthesis of ADC molecules.
    Mal-PEG4-NPV-PABC-DMEDA
  • HY-182990
    N3-Methylcytidine phosphoramidite [5′-O-DMT2′-O-TBDMS-m3 CAc] 2931457-60-0
    N3-Methylcytidine phosphoramidite [5′-O-DMT2′-O-TBDMS-m3 CAc] is a phosphoramidite monomer. Phosphoramidites can be used in the synthesis of oligonucleotides.
    N3-Methylcytidine phosphoramidite [5′-O-DMT2′-O-TBDMS-m3 CAc]
  • HY-182991
    2′-O-Hexyl-adenosine 2642321-62-6 98%
    2′-O-Hexyl-adenosine is a nucleoside derivative that can be used for the synthesis of RNA.
    2′-O-Hexyl-adenosine