1. Cytoskeleton
  2. Integrin
  3. Zaurategrast

Zaurategrast (Synonyms: CT7758)

Cat. No.: HY-70073 Purity: 98.81%
Handling Instructions

Zaurategrast (CT7758) is a potent and oral-effective α4-integrin inhibitor.

For research use only. We do not sell to patients.

Zaurategrast Chemical Structure

Zaurategrast Chemical Structure

CAS No. : 455264-31-0

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply Now  
10 mM * 1 mL in DMSO USD 234 In-stock
Estimated Time of Arrival: December 31
5 mg USD 204 In-stock
Estimated Time of Arrival: December 31
10 mg USD 360 In-stock
Estimated Time of Arrival: December 31
25 mg USD 708 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Description

Zaurategrast (CT7758) is a potent and oral-effective α4-integrin inhibitor[1].

IC50 & Target

α4-integrin[1]

In Vitro

Zaurategrast (CT7758) is a carboxylate containing α4β1/α4/β7 integrin antagonist[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

521.41

Formula

C₂₆H₂₅BrN₄O₃

CAS No.

455264-31-0

SMILES

O=C1C(Br)=C(C12CCCCC2)N[[email protected]](C(O)=O)CC3=CC=C(NC4=NC=CC5=CC=NC=C45)C=C3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (191.79 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.9179 mL 9.5894 mL 19.1788 mL
5 mM 0.3836 mL 1.9179 mL 3.8358 mL
10 mM 0.1918 mL 0.9589 mL 1.9179 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 3.25 mg/mL (6.23 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 3.25 mg/mL (6.23 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
Animal Administration

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

References
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This equation is commonly abbreviated as: C1V1 = C2V2

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Keywords:

ZaurategrastCT7758CT 7758CT-7758IntegrinInhibitorinhibitorinhibit

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Zaurategrast
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