2. GPCR/G Protein
  3. Prostaglandin Receptor
  4. CRTh2 antagonist 1

CRTh2 antagonist 1 is a CRTh2 antagonist with an IC50 of 89 nM.

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CRTh2 antagonist 1

CRTh2 antagonist 1 화학구조

CAS No. : 1379445-54-1

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CRTh2 antagonist 1 Related Antibodies

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제품 설명

CRTh2 antagonist 1 is a CRTh2 antagonist with an IC50 of 89 nM.

IC50 & Target

IC50: 89 nM (CRTh2)[1]
Cellular Effect
Cell Line Type Value Description References
CHO-K1 IC50
89 nM
Compound: 32
Antagonist activity at CRTh2 receptor (unknown origin) overexpressed in CHOK1 cell membranes assessed as inhibition of [35S]-GTPgammaS binding preincubated for 1 hr followed by 50 nM PGD2 and 0.1 nM [35S]-GTPgammaS addition measured after 2 hrs by liquid scintillation counting analysis
Antagonist activity at CRTh2 receptor (unknown origin) overexpressed in CHOK1 cell membranes assessed as inhibition of [35S]-GTPgammaS binding preincubated for 1 hr followed by 50 nM PGD2 and 0.1 nM [35S]-GTPgammaS addition measured after 2 hrs by liquid scintillation counting analysis
[PMID: 23601708]
In Vitro

CRTh2 antagonist 1 is compound 32[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

CRTh2 antagonist 1 Related Antibodies
분자량

455.53

화학식

C23H25N3O5S
CAS No.
SMILES

O=C(O)CC1=C(C)N(CC2=CC=CC=C2S(=O)(N3CCOCC3)=O)N=C1C4=CC=CC=C4
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
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CRTh2 antagonist 1 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CRTh2 antagonist 11379445-54-1Prostaglandin ReceptorInhibitorinhibitorinhibit

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상품명:
CRTh2 antagonist 1
Cat. No.:
HY-112265
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