2. Others

Others

Others

Related Products

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There are a number of inhibitors, agonists, and antagonists which we cannot make precise classification because the research area is still unknown.

Others Related Products (73826):

Cat. No. Product Name CAS No. Purity Chemical Structure
  • HY-142907S
    (2-Fluoro-4-biphenyl)acetic acid-d5 2733149-72-7 99.64%
    (2-Fluoro-4-biphenyl)acetic acid-d5 is the deuterium labeled (2-Fluoro-4-biphenyl)acetic acid.
    (2-Fluoro-4-biphenyl)acetic acid-d5
  • HY-143645S
    Glycochenodeoxycholic acid 3-sulfate-d5 disodium 99.33%
    Glycochenodeoxycholic acid 3-sulfate-d5 (disodium) is the deuterium labeled Glycochenodeoxycholic acid 3-sulfate disodium.
    Glycochenodeoxycholic acid 3-sulfate-d5 disodium
  • HY-143824S
    Malachite green-d5 (picrate) 1258668-21-1 99.00%
    Malachite green-d5 (picrate) is the deuterium labeled Malachite green picrate.
    Malachite green-d5 (picrate)
  • HY-143915S
    Amitriptyline-N-glucuronide-d3
    Amitriptyline-N-glucuronide-d3 is the deuterium labeled Amitriptyline-N-glucuronide.
    Amitriptyline-N-glucuronide-d3
  • HY-143922S
    N-Desmethyl Bedaquiline-d6 2271264-26-5
    N-Desmethyl Bedaquiline-d6 is the deuterium labeled N-Desmethyl Bedaquiline.
    N-Desmethyl Bedaquiline-d6
  • HY-143979S
    1-(2-Chloroethyl)-3-((1R,4R)-4-hydroxycyclohexyl)-1-nitrosourea-d4 99.0%
    trans-4’-Hydroxy CCNU Lomustine-d4 is the deuterium labeled trans-4’-Hydroxy CCNU Lomustine.
    1-(2-Chloroethyl)-3-((1R,4R)-4-hydroxycyclohexyl)-1-nitrosourea-d4
  • HY-144008B
    C8 PEG750 Ceramide 212116-76-2 99.94%
    C8 PEG750 Ceramide is a lipid product. C8 PEG750 Ceramide synthesizes a lipid bilayer carrier for the selective delivery of various diagnostic and therapeutic agents to acidic diseased cells.
    C8 PEG750 Ceramide
  • HY-144012A
    DPPE-PEG350 474922-84-4 99%
    DPPE-PEG350 is a CD1d-dependent lipid antagonist thus blocking the ERK phosphorylation pathway in iNKT cells. DPPE-PEG350 is a PEG lipid functional end group used in the synthesis of liposomes (LPs) for the design of conjugated polymer nanoparticles.
    DPPE-PEG350
  • HY-144012H
    DPPE-PEG5000 474922-84-4 99.94%
    DPPE-PEG5000 (16:0 PEG5000 PE) is a polymer-lipid conjugate and LipoParticle stabilizer with a PEG chain of 5,000 g/mol molecular weight attached to its polar head, and it can be internalized by biological membranes. DPPE-PEG5000 enables LipoParticle to maintain colloidal stability after 20-fold dilution in PBS or cell culture medium, and prevents aggregate formation during lyophilization and rehydration. DPPE-PEG5000 helps enhance the non-cytotoxic property of LipoParticle formulations against human osteoblasts. DPPE-PEG5000 serves as a PEG lipid functional end group for synthesizing liposomes (LPs), is used in the design of conjugated polymer nanoparticles, and applies to research related to bone and joint infections.
    DPPE-PEG5000
  • HY-144140S
    4-Nitroso hydrochlorothiazide-13C,15N2,d2 99.34%
    4-Nitroso hydrochlorothiazide-13C,15N2,d2 is the deuterium, 13C-, and 15-labeled 4-Nitroso hydrochlorothiazide.
    4-Nitroso hydrochlorothiazide-13C,15N2,d2
  • HY-144247S
    Edaravone glucuronide-d5 sodium 99.9%
    Edaravone glucuronide-d5 (sodium) is the deuterium labeled Edaravone glucuronide sodium.
    Edaravone glucuronide-d5 sodium
  • HY-144427S
    Vitamin E-13C2,d6 2483824-69-5 98.0%
    Vitamin E-13C2,d6 is a 13C-labeled and deuterium labeled Vitamin E.
    Vitamin E-13C2,d6
  • HY-145008S
    (±)9(10)-DiHOME-d4 1215168-76-5 ≥99.0%
    (±)9(10)-DiHOME-d4 is the deuterium labeled (±)9(10)-DiHOME.
    (±)9(10)-DiHOME-d4
  • HY-145576B
    2-Amino-8-oxononanoic acid hydrochloride 2984160-77-0 98.0%
    2-Amino-8-oxononanoic acid (hydrochloride) is the hydrochloride form of 2-Amino-8-oxononanoic acid. 2-Amino-8-oxononanoic acid is an amino acid, incorporation into proteins in E.coli in genetic. 2-Amino-8-oxononanoic acid is efficient in labeling of proteins with different probes with a site-specific manner under a mild condition close to the physiological pH.
    2-Amino-8-oxononanoic acid hydrochloride
  • HY-146066A
    (R)-α7 nAchR-JAK2-STAT3 agonist 1 99.59%
    (R)-α7 nAchR-JAK2-STAT3 agonist 1 is the R-enantiomer of α7 nAchR-JAK2-STAT3 agonist 1 (HY-146066). α7 nAchR-JAK2-STAT3 agonist 1 is a potent α7 nAchR-JAK2-STAT3 agonist, with an IC50 value of 0.32 μM for nitric oxide (NO). α7 nAchR-JAK2-STAT3 agonist 1 effectively suppresses the expression of iNOS, IL-1β, and IL-6 in murine RAW264.7 macrophages. α7 nAchR-JAK2-STAT3 agonist 1 can inhibit LPS-induced NO release, NF-κB activation and cytokine production. α7 nAchR-JAK2-STAT3 can be used for researching sepsis.
    (R)-α7 nAchR-JAK2-STAT3 agonist 1
  • HY-146241B
    SN40 hydrochloride 2768663-15-4 98.00%
    SN40 hydrochloride is a potent amino acid transport (AAT) inhibitor with Kis of 7.29 μM, 2.42 μM, 2.94 μM, 5.55 μM, 24.43 μM and 5.55 μM for rat ASCT2, human ASCT2, EAAT1, EAAT2, EAAC1 and EAAT5, respectively. SN40 hydrochloride can be used for researching anticancer.
    SN40 hydrochloride
  • HY-146248A
    TFMU-ADPr triethylamine
    TFMU-ADPr triethylamine is a selective reporter substrate of SARS-CoV-2 Macro1 (IC50=0.59 μM), with an excitation wavelength (λEx) of 385 nm, and an emission wavelength (λEm) of 502 nm (or 495 nm). TFMU-ADPr triethylamine can also undergo enzymatic hydrolysis with Poly(ADP-ribose) Glycohydrolase (PARG) sourced from human, Tetrahymena thermophila and ADP-ribosylhydrolase 3 from human to release fluorophores, thereby directly reporting total poly (ADP-ribose) hydrolase activity. TFMU-ADPr triethylamine binds to the ADPr-binding site of SARS-CoV-2 Macro1, and its TFMU moiety inserts into the narrow hydrophobic groove of this protein. TFMU-ADPr triethylamine can thus be used to evaluate small-molecule inhibitors targeting PAR hydrolases under in vitro conditions, to investigate the regulatory mechanisms of ADP-ribosyl catabolic enzymes, or to detect PAR hydrolase activity in whole-cell lysate assays. TFMU-ADPr triethylamine is also applicable to COVID-19-related research.
    TFMU-ADPr triethylamine
  • HY-146534S
    Diazinon-d10 100155-47-3
    Diazinon-d10 is the deuterium labeled Diazinon.
    Diazinon-d10
  • HY-146567S
    meso-Erythritol-d6 2714435-98-8 99.9%
    meso-Erythritol-d6 is the deuterium labeled meso-Erythritol (HY-100551). meso-Erythritol is a sugar alcohol that found in a variety of foods (e.g., pear, watermelon), is 60-80% as sweet as sucrose, and can be used as low-calorie sweetener food additives.
    meso-Erythritol-d6
  • HY-146712S
    N-(4-Hydroxyphenyl)acetamide sulfate-d3 sodium 2733160-80-8 98%
    N-(4-Hydroxyphenyl)acetamide sulfate-d3 (sodium) is the deuterium labeled N-(4-Hydroxyphenyl)acetamide sulfate.
    N-(4-Hydroxyphenyl)acetamide sulfate-d3 sodium