1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. 5-HT Receptor
  4. 5-HT4 Receptor Inhibitors

5-HT4 Receptor Inhibitors

5-HT1 Receptor

5-HT2 Receptor

5-HT3 Receptor

5-HT5 Receptor

5-HT6 Receptor

5-HT7 Receptor

5-HT Receptor

5-HT4 Receptor

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform 5-HT4 Receptor together.

Please try each isoform separately.

5-HT4 Receptor Specific Inhibitors, Agonists, Antagonists & Modulators
Product Name 5-HT4 Receptor 5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT4 Receptor Selectivity Purity
Cisapride
5-HT4 Receptor, EC50: 0.14 μM
          Selective Agonist 99.72%
Piboserod
5-HT4 Receptor
          Selective Antagonist 99.12%
Mosapride citrate
5-HT4 Receptor
          Selective Agonist 99.80%
PF-04995274
5-HT4 Receptor
          Selective Agonist 99.42%
Velusetrag
5-HT4 Receptor, pKi: 7.7
          Selective Agonist 99.64%
Velusetrag hydrochloride
5-HT4 Receptor, pKi: 7.7
          Selective Agonist 96.65%
GR 113808
5-HT4 Receptor
5-HT1A Receptor
5-HT2A Receptor
5-HT2C Receptor
5-HT3 Receptor
    Selective Antagonist ≥98.0%
Mosapride
5-HT4 Receptor
          Selective Agonist
Revexepride
5-HT4 Receptor
          Selective Agonist 95.81%
Felcisetrag
huamn 5-HT4(c) Receptor, pKi: 9.4
          Selective Agonist 99.65%
ML 10302 hydrochloride
5-HT4 Receptor, EC50: 4 nM
5-HT4 Receptor, Ki: 1.07 nM
   
5-HT3 Receptor, Ki: 782 nM
    Selective Agonist
Renzapride
5-HT4 Receptor, Ki: 115 nM
          Selective Agonist
Piboserod hydrochloride
5-HT4 Receptor
          Selective Antagonist
MHP 133
5-HT4 Receptor
          Selective Inhibitor
Tegaserod maleate
5-HT4 Receptor (Agonist)
 
5-HT2B Receptor (Antagonist)
      Pan Modulator 99.75%
Prucalopride
5-HT4A Receptor, pKi: 8.6
5-HT4B Receptor, pKi: 8.1
          Pan Agonist 99.89%
SB 271046 Hydrochloride
5-HT4 Receptor, pKi: 5.27
5-HT1D Receptor, pKi: 6.55
5-HT1A Receptor, pKi: 6.35
5-HT1B Receptor, pKi: 6.05
5-HT1F Receptor, pKi: 5.95
5-HT1E Receptor, pKi: <4.99
5-HT2A Receptor, pKi: 5.62
5-HT2B Receptor, pKi: 5.41
Human 5-HT2C Receptor, pKi: 5.73
 
5-HT6 Receptor, pKi: 8.92-9.02
5-HT7 Receptor, pKi: 5.39
Pan Antagonist 98.64%
Prucalopride succinate
5-HT4A Receptor, pKi: 8.6
5-HT4B Receptor, pKi: 8.1
          Pan Agonist 99.83%
Fabesetron
5-HT4 Receptor
   
5-HT3 Receptor
    Pan Antagonist 95.72%
Relenopride hydrochloride
5-HT4 Receptor, Ki: 4.96 nM
 
5-HT2A Receptor, Ki: 600 nM
5-HT2B Receptor, Ki: 31 nM
5-HT2B Receptor, IC50: 2.1 μM
      Pan Agonist 99.13%
Lintopride
5-HT4 Receptor
   
5-HT3 Receptor
    Pan Antagonist 96.38%
(±)-Fabesetron hydrochloride
5-HT4 Receptor
   
5-HT3 Receptor
    Pan Antagonist
BIMU 8
5-HT4 Receptor, EC50: 18 nM
          Pan Agonist
5-HT4 antagonist 1
5-HT4 Receptor, pKi: 9.6
          Pan Antagonist
Sulamserod
5-HT4 Receptor
          Pan Antagonist