Capeserod hydrochloride
Capeserod hydrochloride (SL65.0155) is a 5-HT4(e) receptor partial agonist (Ki=0.6 nM) with potent cognitive enhancing properties. Capeserod hydrochloride acts as a partial agonist in cells expressing 5-HT4(b) and 5-HT4(e) splice variants, stimulating cAMP production with IC50 values of 244 and 29 nM, respectively. Capeserod hydrochloride is used in the study of memory impairment and dementia.
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- CAS No.: 191023-43-5
- Formule: C23H26Cl2N4O4
- Masse moléculaire:493.38
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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5-HT4(e) Receptor |
5-HT4B Receptor |
5-HT4(e) Receptor 0.6 nM (Ki) |
Chemical Information
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CAS No. 191023-43-5
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Masse moléculaire 493.38
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Formule C23H26Cl2N4O4
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SMILES
O=C1OC(C2=C3OCCOC3=C(N)C(Cl)=C2)=NN1C4CCN(CC4)CCC5=CC=CC=C5.Cl
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Synonyms
SL65.0155
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)