1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. 5-HT Receptor
  4. 5-HT Receptor Isoform

5-HT Receptor


5-HT Receptor Related Products (199):

Cat. No. Product Name Effect Purity
  • HY-12560A
    Antagonist 99.70%
    PNU-282987 is a potent α7 nicotinic acetylcholine receptor (nAChR) agonist with an EC50 of 154 nM.
  • HY-B0670A
    Dihydroergotamine mesylate
    Agonist 99.98%
    Dihydroergotamine mesylate is an ergot alkaloid used to treat migraines.
  • HY-B0965
    Thioridazine hydrochloride
    Antagonist 99.96%
    Thioridazine hydrochloride, an orally active antagonist of the dopamine receptor D2 family proteins, exhibits potent anti-psychotic and anti-anxiety activities.
  • HY-B1115
    Buspirone hydrochloride
    Agonist 99.99%
    Buspirone hydrochloride is a 5-HT1A receptor agonist.
  • HY-B0478
    Trazodone hydrochloride
    Antagonist 99.87%
    Trazodone (hydrochloride) (AF-1161) is an antidepressant belonging to the class of serotonin receptor antagonists and reuptake inhibitors for treatment of anxiety disorders.
  • HY-101456
    PCPA methyl ester hydrochloride
    Inhibitor 99.89%
    PCPA methyl ester hydrochloride (4-Chloro-DL-phenylalanine methyl ester hydrochloride), a reversible tryptophan hydroxylase inhibitor, is a serotonin (5-HT) synthesis inhibitor.
  • HY-107613
    R 59-022
    Antagonist 99.82%
    R 59-022 (DKGI-I) is a DGK inhibitor (IC50: 2.8 µM).
  • HY-B1693
    Antagonist 99.98%
    Levomepromazine (Methotrimeprazine) is an orally available neuroleptic agent, which is commonly used to relieve nausea and vomiting in palliative care settings.
  • HY-P1422A
    Spadin TFA
    Inducer 99.73%
    Spadin TFA, a natural peptide derived from a propeptide released in blood, is a potent TREK-1 channel blocker with an IC50 value of 10 nM.
  • HY-14537
    Latrepirdine dihydrochloride
    Antagonist 99.71%
    Latrepirdine dihydrochloride is a neuroactive compound with antagonist activity at histaminergic, α-adrenergic, and serotonergic receptors.
  • HY-108324
    Antagonist 99.76%
    (Z)-Thiothixene is an antagonist of serotonergic receptor extracted from patent US 20150141345 A1.
  • HY-30152
    Antagonist 99.75%
    Xanthotoxol (8-Hydroxypsoralen) is a biologically active linear furocoumarin, shows strong pharmacological activities as anti-inflammatory, antioxidant, 5-HT antagonistic, and neuroprotective effects.
  • HY-112390A
    Syk Inhibitor II
    Inhibitor 98.05%
    Syk Inhibitor II is a potent, high selective and ATP-competitive Syk inhibitor with an IC50 of 41 nM.
  • HY-B1371
    Spiperone is a potent dopamine D2, serotonin 5-HT1A, and serotonin 5-HT2A antagonist.
  • HY-B0740
    Cyclobenzaprine hydrochloride
    Antagonist 99.91%
    Cyclobenzaprine hydrochloride (MK130 hydrochloride) is a skeletal muscle relaxant and a central nervous system (CNS) depressant.
  • HY-16978
    Antagonist 99.92%
    TG6-10-1 is an EP2 antagonist, shows low-nanomolar antagonist activity against only EP2, >300-fold selectivity over human EP3, EP4, and IP receptors, 100-fold selectivity over EP1 receptors.
  • HY-123205
    Inhibitor 99.47%
    Oxatomide is a potent and orally active dual H1-histamine receptor and P2X7 receptor antagonist with antihistamine and anti-allergic activity.
  • HY-102064
    SR 57227A
    Agonist 99.57%
    SR 57227A is a potent, orally active and selective 5-HT3 receptor agonist, with ability to cross the blood brain barrier.
  • HY-N0749A
    Jatrorrhizine hydroxide
    Inhibitor 98.02%
    Jatrorrhizine hydroxide is an alkaloid isolated from Coptis chinensis with neuroprotective, antimicrobial, antiplasmodial and antioxidant activities.
  • HY-U00096
    Ansofaxine hydrochloride
    Inhibitor 99.87%
    Ansofaxine hydrochloride (LY03005; LPM570065) is a triple reuptake inhibitor; inhibits serotonin, dopamine and norepinephrine reuptake with IC50 values of 723, 491 and 763 nM, respectively.