5-HT Receptor

5-HT Receptor Related Products (199):

By Type:	Pan (22) Selective (2)
By Effects:	Inhibitors (33) Agonists (43) Antagonists (76) Activator (1) Modulators (11) Inducers (2)

Cat. No.	Product Name	Effect	Purity

HY-12560A

PNU-282987	Antagonist	99.70%
PNU-282987 is a potent α7 nicotinic acetylcholine receptor (nAChR) agonist with an EC₅₀ of 154 nM.

HY-B0670A

Dihydroergotamine mesylate	Agonist	99.98%
Dihydroergotamine mesylate is an ergot alkaloid used to treat migraines.

HY-B0965

Thioridazine hydrochloride	Antagonist	99.96%
Thioridazine hydrochloride, an orally active antagonist of the dopamine receptor D2 family proteins, exhibits potent anti-psychotic and anti-anxiety activities.

HY-B1115

Buspirone hydrochloride	Agonist	99.99%
Buspirone hydrochloride is a 5-HT1A receptor agonist.

HY-B0478

Trazodone hydrochloride	Antagonist	99.87%
Trazodone (hydrochloride) (AF-1161) is an antidepressant belonging to the class of serotonin receptor antagonists and reuptake inhibitors for treatment of anxiety disorders.

HY-101456

PCPA methyl ester hydrochloride	Inhibitor	99.89%
PCPA methyl ester hydrochloride (4-Chloro-DL-phenylalanine methyl ester hydrochloride), a reversible tryptophan hydroxylase inhibitor, is a serotonin (5-HT) synthesis inhibitor.

HY-107613

R 59-022	Antagonist	99.82%
R 59-022 (DKGI-I) is a DGK inhibitor (IC₅₀: 2.8 µM).

HY-B1693

Levomepromazine	Antagonist	99.98%
Levomepromazine (Methotrimeprazine) is an orally available neuroleptic agent, which is commonly used to relieve nausea and vomiting in palliative care settings.

HY-P1422A

Spadin TFA	Inducer	99.73%
Spadin TFA, a natural peptide derived from a propeptide released in blood, is a potent TREK-1 channel blocker with an IC₅₀ value of 10 nM.

HY-14537

Latrepirdine dihydrochloride	Antagonist	99.71%
Latrepirdine dihydrochloride is a neuroactive compound with antagonist activity at histaminergic, α-adrenergic, and serotonergic receptors.

HY-108324

(Z)-Thiothixene	Antagonist	99.76%
(Z)-Thiothixene is an antagonist of serotonergic receptor extracted from patent US 20150141345 A1.

HY-30152

Xanthotoxol	Antagonist	99.75%
Xanthotoxol (8-Hydroxypsoralen) is a biologically active linear furocoumarin, shows strong pharmacological activities as anti-inflammatory, antioxidant, 5-HT antagonistic, and neuroprotective effects.

HY-112390A

Syk Inhibitor II	Inhibitor	98.05%
Syk Inhibitor II is a potent, high selective and ATP-competitive Syk inhibitor with an IC₅₀ of 41 nM.

HY-B1371

Spiperone	Antagonist
Spiperone is a potent dopamine D2, serotonin 5-HT_1A, and serotonin 5-HT_2A antagonist.

HY-B0740

Cyclobenzaprine hydrochloride	Antagonist	99.91%
Cyclobenzaprine hydrochloride (MK130 hydrochloride) is a skeletal muscle relaxant and a central nervous system (CNS) depressant.

HY-16978

TG6-10-1	Antagonist	99.92%
TG6-10-1 is an EP2 antagonist, shows low-nanomolar antagonist activity against only EP2, >300-fold selectivity over human EP3, EP4, and IP receptors, 100-fold selectivity over EP1 receptors.

HY-123205

Oxatomide	Inhibitor	99.47%
Oxatomide is a potent and orally active dual H1-histamine receptor and P2X7 receptor antagonist with antihistamine and anti-allergic activity.

HY-102064

SR 57227A	Agonist	99.57%
SR 57227A is a potent, orally active and selective 5-HT3 receptor agonist, with ability to cross the blood brain barrier.

HY-N0749A

Jatrorrhizine hydroxide	Inhibitor	98.02%
Jatrorrhizine hydroxide is an alkaloid isolated from Coptis chinensis with neuroprotective, antimicrobial, antiplasmodial and antioxidant activities.

HY-U00096

Ansofaxine hydrochloride	Inhibitor	99.87%
Ansofaxine hydrochloride (LY03005; LPM570065) is a triple reuptake inhibitor; inhibits serotonin, dopamine and norepinephrine reuptake with IC₅₀ values of 723, 491 and 763 nM, respectively.

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