2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. SC-53606

SC-53606 is a potent and selective 5-HT4 receptor antagonist, with a pA2 value of 8.13. SC-53606 acts as an antagonist of 5-HT4 receptor-mediated relaxation of Carbachol (HY-B1208)-induced contractions.

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SC-53606

SC-53606 Chemical Structure

CAS No. : 151898-33-8

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SC-53606 Related Antibodies

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Description

SC-53606 is a potent and selective 5-HT4 receptor antagonist, with a pA2 value of 8.13. SC-53606 acts as an antagonist of 5-HT4 receptor-mediated relaxation of Carbachol (HY-B1208)-induced contractions[1][2].

IC50 & Target[1][2]

5-HT4 Receptor

 

Molecular Weight

318.80

Formula

C16H19ClN4O
CAS No.
SMILES

O=C(NC[C@H]1[C@@]2(CCCN2CC1)[H])C3=CC(Cl)=CN4C3=NC=C4
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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SC-53606 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SC-53606151898-33-8SC53606SC 536065-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorcontractionsInhibitorinhibitorinhibit

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