1. Signaling Pathways
  2. Others
  3. Estrogen Receptor/ERR
  4. Estrogen receptor Isoform
  5. Estrogen receptor Antagonist

Estrogen receptor Antagonist

Estrogen receptor Antagonists (3):

Cat. No. Product Name Effect Purity
  • HY-109176
    Giredestrant
    Antagonist 99.52%
    Giredestrant (GDC-9545), a non-steroidal estrogen receptor (ER) ligand, is an orally active and selective ER antagonist.
  • HY-135903
    Giredestrant tartrate
    Antagonist
    Giredestrant tartrate (GDC-9545 tartrate), a non-steroidal ER ligand, is an orally active and selective estrogen receptor (ER) antagonist.
  • HY-143439
    LX-039
    Antagonist
    LX-039 is a highly potent, selective and orally active estrogen receptor degrader with EC50 value of 2.29 nM.