1. Signaling Pathways
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  3. Estrogen Receptor/ERR
  4. Estrogen receptor Isoform

Estrogen receptor

 

Estrogen receptor Related Products (15):

Cat. No. Product Name Effect Purity
  • HY-13757A
    Tamoxifen
    Modulator 99.92%
    Tamoxifen (ICI 47699) is an orally active, selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells.
  • HY-16950
    4-Hydroxytamoxifen
    Modulator 99.96%
    4-Hydroxytamoxifen ((Z)-4-Hydroxytamoxifen) is an orally active, selective estrogen receptor modulator (SERM).
  • HY-13757
    Tamoxifen Citrate
    Modulator 99.93%
    Tamoxifen Citrate (ICI 46474) is an orally active, selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells.
  • HY-109176
    Giredestrant
    Antagonist 99.52%
    Giredestrant (GDC-9545), a non-steroidal estrogen receptor (ER) ligand, is an orally active and selective ER antagonist.
  • HY-16950A
    (E/Z)-4-Hydroxytamoxifen
    Modulator 99.60%
    (E/Z)-4-Hydroxytamoxifen (Afimoxifene) is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers.
  • HY-N6678
    Zearalanone
    Activator 98.11%
    Zearalenone is a nonsteroidal estrogenic mycotoxin produced by Fusarium species, which colonizes several grains.
  • HY-135309
    PROTAC ER Degrader-4
    Inhibitor 98.05%
    PROTAC ER Degrader-4 is a von Hippel-Lindau-based PROATC estrogen receptor (ER) degrader, binding to ER with an IC50 of 0.8 nM.
  • HY-13757AS
    Tamoxifen-​d5
    Modulator 99.77%
    Tamoxifen-d5 (ICI 47699-d5) is a deuterium labeled Tamoxifen.
  • HY-135903
    Giredestrant tartrate
    Antagonist
    Giredestrant tartrate (GDC-9545 tartrate), a non-steroidal ER ligand, is an orally active and selective estrogen receptor (ER) antagonist.
  • HY-N8170
    4',2-Dihydroxy-4,6-dimethoxydihydrochalcone
    Agonist
    4',2-Dihydroxy-4,6-dimethoxydihydrochalcone, an estrogen agonist, shows binding affinity for bovine uterine estrogen receptor with an IC5050 of 15 μM.
  • HY-16950B
    (E)-4-Hydroxytamoxifen
    Modulator 98.27%
    (E)-4-Hydroxytamoxifen ((E)-Afimoxifene), the less active isomer of (Z)-4-hydroxytamoxifen, is an estrogen receptor modulator.
  • HY-143439
    LX-039
    Antagonist
    LX-039 is a highly potent, selective and orally active estrogen receptor degrader with EC50 value of 2.29 nM.
  • HY-13738
    Raloxifene
    Modulator
    Raloxifene (Keoxifene) is a benzothiophene-derived selective estrogen receptor modulator (SERM).
  • HY-116896
    LY117018
    Modulator
    LY117018, a Raloxifene analog, is a selective estrogen receptor modulator.
  • HY-113251
    2-Hydroxyestrone
    2-Hydroxyestrone (Catecholestrone) is a specific receptor-mediated antiestrogenic agent.