43 Results for "

amide analogs

" in MedChemExpress (MCE) Product Catalog:
Products (43)

43 Results for "amide analogs" in MCE Product Catalog:

  • Targets Recommended:
Cat. No.: HY-103423
CAS No.: 114200-31-6
Purity:  98.09%
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

PAOPA, an analog of L-proline-l-leucine-glycine amide (PLG) peptide, is an allosteric modulator of Dopamine D2 Receptor. PAOPA can effectively reduce behavioral abnormalities in rodent models of schizophrenia. PAOPA increases the high affinity dopamine D2 receptor and promotes its binding to agonists .
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Cat. No.: HY-108490
CAS No.: 449173-19-7
Purity:  99.20%
Target:  

LPL Receptor

Research Areas:  

Inflammation/Immunology

VPC 23019, an aryl amide-containing Sphingosine 1-phosphate (S1P) analog, is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively) and an agonist at the S1P4 and S1P5 receptors (pEC50= 6.58 and 7.07, respectively) .
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Cat. No.: HY-W008213
CAS No.: 6342-60-5
2-Chloro-5-methylbenzoic acid can be used to synthesize amide when coupled with 1-Adamantylmethanamine. 2-Chloro-5-methylbenzoic acid can also give analog when coupled with an amine using EDC hydrochlorie and Et3N in anhydrous CH2Cl2 .
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Cat. No.: HY-P3594
CAS No.: 94034-78-3
Target:  

GHR

Research Areas:  

Endocrinology

[His1,Nle27] GHRF (1-32), amide, human is a Growth hormone releasing hormone (GHRH) analog. [His1,Nle27] GHRF (1-32), amide, human has great receptor affinity for GHRHR .
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Cat. No.: HY-161943
CAS No.: 3094051-91-6
Target:  

Influenza Virus

Research Areas:  

Neurological Disease

NEU3-IN-1 (compound 963) is a NEU3 inhibitor (Ki: 0.12 μM; IC50: 0.31 μM) based on the 2-deoxy-2,3-didehydro-N-acetylneuraminic acid (DANA) scaffold and is a C9 biphenylcarbamate derivative. NEU is a human neuraminidase with 4 isozymes; NEU3-IN-1 is an important tool for studying the function of NEU3 isozymes; its amide and triazole linker analogs are selective for NEU1 and NEU4 isozymes, respectively .
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Cat. No.: HY-151821
CAS No.: 2566404-75-7
Target:  

ADC Linkers

Research Areas:  

Others

Sulfo DBCO-PEG3-acid is a click chemistry reagent containing an azide group. Sulfo DBCO-PEG3-acid is an analog of DBCO-Acid with PEG linker and a DBCO group. The DBCO groups is commonly used for copper-free Click Chemistry reactions due to its strain promoted high energy. The hydrophilic PEG chain and sulfo group increase water solubility. The terminal carboxylic acid can react with primary amine groups in the presence of activators (e.g. EDC, or HATU) to form a stable amide bond. Reagent grade, for research use only .
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Cat. No.: HY-137462
CAS No.: 38678-60-3
Synonyms: L-Leucyl-L-phenylalaninamide
Leucyl-phenylalanine amide (L-Leucyl-L-phenylalaninamide) is a dipeptide analog. Leucyl-phenylalanine amide is a ligand of SP1-7 with a Ki value of 10.2 nM. Leucyl-phenylalanine amide shows no binding activity to human NK-1 or NK-3 receptors .
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Cat. No.: HY-44630
CAS No.: 2172819-75-7
Synonyms: (S,R,S)-AHPC-CO-C6-COOH
Research Areas:  

Cancer

VH 032 amide-alkylC6-acid ((S,R,S)-AHPC-CO-C6-COOH) is a VH032 analog that acts as a ligand for VHL, recruiting von Hippel-Lindau (VHL) protein. VH 032 amide-alkylC6-acid can be used in the synthesis of PROTACs .
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Cat. No.: HY-114867
CAS No.: 1163135-92-9
Synonyms: 15(R)-17-phenyl trinor PGF2α ethyl amide
Research Areas:  

Endocrinology

(15R)-Bimatoprost (15(R)-17-phenyl trinor PGF2α ethyl amide) is a prostaglandin analog used to study glaucoma and ocular hypertension. (15R)-Bimatoprost is an isomer of Bimatoprost with an inverted (β) hydroxyl group on C-15 .
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Cat. No.: HY-P4555
CAS No.: 340821-13-8
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide (Compound 4) is a somatostatin analog with Kds of 0.61, 11.05, 23.5, 1200 and >1000 nM for SSTR5, SSTR3, SSTR2, SSTR1 and SSTR4, respectively .
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Cat. No.: HY-151820
CAS No.: 2765066-36-0
Purity:  95.12%
Target:  

ADC Linkers

Research Areas:  

Others

DBCO-PEG24-acid is a click chemistry reagent. DBCO-PEG24-acid is an analog of DBCO-Acid with PEG linker and a DBCO group. The DBCO groups is commonly used for copper-free Click Chemistry reactions due to its strain promoted high energy. The hydrophilic PEG chain allows for increased water solubility. The terminal carboxylic acid can react with primary amine groups in the presence of activators (e.g. EDC, or HATU) to form a stable amide bond. Reagent grade, for research use only .
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Cat. No.: HY-148840
Research Areas:  

Others

Sulfo DBCO-PEG3-NHS ester is a click chemistry reagent containing an azide group. Sulfo DBCO-PEG3-NHS ester is an analog of DBCO-Acid with PEG linker and a DBCO group. The DBCO group is commonly used for copper-free Click Chemistry reactions due to its strain promoted high energy. The hydrophilic PEG chain and sulfo group increase water solubility. The terminal carboxylic acid can react with primary amine groups in the presence of activators (e.g. EDC, or HATU) to form a stable amide bond. Reagent grade, for research use only .
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Cat. No.: HY-P4818
CAS No.: 173833-08-4
Research Areas:  

Metabolic Disease

Human PTH-(1-31) amide is a PTH analog. Human PTH-(1-31) amide stimulate phosphatidylcholine hydrolysis and stimulates adenylyl cyclase release .
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Cat. No.: HY-120467
CAS No.: 1175838-84-2
Synonyms: Bimatoprost serinol amide
Research Areas:  

Endocrinology

Bima SA (Bimatoprost serinol amide) is a Prostaglandin analog and has the potential for the research of glaucoma .
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Cat. No.: HY-W746888
CAS No.: 1176637-26-5
Synonyms: 17-p-PGF2α-NEt2; 17-Phenyl trinor PGF2α diethyl amide
Research Areas:  

Cardiovascular Disease

17-Phenyl trinor prostaglandin F2α diethyl amide (17-phenyl trinor PGF2α diethyl amide) is a PGF analog with hypotensive efficacy .
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Cat. No.: HY-118599
CAS No.: 54130-36-8
Research Areas:  

Others

Prostaglandin F2α ethyl amide is an analog of Prostaglandin F2α (HY-12956). Prostaglandin F2α ethyl amide is supposed to be potent lowering intraocular pressure (IOP) for its N-ethyl amide group, like Bimatoprost (HY-B0191) .
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Cat. No.: HY-176021
Research Areas:  

Cardiovascular Disease

U-44069 serinol amide is a derivative of U-44069 (HY-121825). U-44069 serinol amide is a stable analog of the endoperoxide prostaglandin H2 (HY-136500). U-44069 serinol amide is a vasoconstrictor that can induce preglomerular Ca 2+ influx .
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Cat. No.: HY-176022
Research Areas:  

Cardiovascular Disease

U-46619 serinol amide is a derivative of U-46619 (HY-108566). U-46619 serinol amide is a stable analog of Thromboxane A2 (HY-113350) (TXA2). U-46619 serinol amide is a potent TXA2 agonist that can induce platelet shape change and aggregation .
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Cat. No.: HY-P10309
CAS No.: 120527-89-1
Synonyms: [Nle8'18,Tyr34]hPTH (3-34) amide
Target:  

PTHR

Research Areas:  

Endocrinology

[Nle8,18,Tyr34]-pTH (3-34) amide human ([Nle8,18,Tyr34]hPTH (3-34) amide) is a parathyroid hormone (PTH) analog .
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Cat. No.: HY-124219
CAS No.: 1421369-12-1
Synonyms: 17-Phenoxy trinor PGF2α ethyl amide
Research Areas:  

Others

17-Phenoxy trinor prostaglandin F2α ethyl amide (17-Phenoxy trinor PGF2α ethyl amide) is an analog of Bimatoprost (HY-12956). 17-Phenoxy trinor prostaglandin F2α ethyl amide is an agonist for Prostaglandin F2α Receptor (FP receptor). 17-Phenoxy trinor prostaglandin F2α ethyl amide is potent to reduce the intraocular pressure and attenuate the glaucoma .
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