FMJ-01-042
FMJ-01-042 is a blood-brain barrier-permeable, low-efficacy partial agonist with high affinity (Kᵢ = 4.33 nM) and exceptional subtype selectivity for the dopamine D4 receptor. FMJ-01-042 exhibits good metabolic stability and is suitable for research on neurological and psychiatric disorders.
Para uso exclusivo en investigación. No vendemos a pacientes.
- Fòrmula: C24H25N5
- Peso molecular:383.49
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Actividad biológica
-
Chemical Information
- Pureza y Documentación
- Referencias
-
Help & FAQs
Ver todos los productos específicos de isoformas Dopamine Receptor
More
Actividad biológica
Descripciòn
In Vitro
FMJ-01-042 (Compound 18) (90 min) can act as a D4R-mediated β-arrestin recruitment antagonist[1].
FMJ-01-042 exhibited good metabolic stability in rat liver microsomes, with a t1/2 value of 56.77 min[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
Peso molecular 383.49
-
Fòrmula C24H25N5
-
SMILES
CC1=CC(N2N=NC(CN3CCN(C4=C5C=CC=CC5=CC=C4)CC3)=C2)=CC=C1
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
FMJ-01-042 Related Classifications
HY-181047 Related Classifications
Powered by Bioz