2. Metabolic Enzyme/Protease Vitamin D Related/Nuclear Receptor
  3. RAR/RXR
  4. RXR antagonist 5

RXR antagonist 5 (compound 22) is a selective retinoic acid X receptor (RXR) antagonist with binding potential to RXR evaluated by modeling.

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RXR antagonist 5

RXR antagonist 5 Chemische Struktur

CAS. Nr. : 1807740-94-8

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Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO
ready for reconstitution
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Solution
10 mM * 1 mL in DMSO Auf Lager
Solid
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RXR antagonist 5 Related Antibodies

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Alle RAR/RXR Isoform-spezifische Produkte anzeigen:

Alle Isoformen anzeigen
RXRα RXRβ RXRγ

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Beschreibung

RXR antagonist 5 (compound 22) is a selective retinoic acid X receptor (RXR) antagonist with binding potential to RXR evaluated by modeling.

Molekulargewicht

366.50

Formel

C23H30N2O2
CAS. Nr.
Appearance

Solid

Color

White to off-white

SMILES

O=C(C1=CN=C(N(CC)C2=C(C)C=C(C(C)(CCC3(C)C)C)C3=C2)C=C1)O
Versand

Room temperature in continental US; may vary elsewhere.
Speicherung
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Lösungsmittel & Löslichkeit
In Vitro: 

DMSO : 50 mg/mL (136.43 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.7285 mL 13.6426 mL 27.2851 mL
5 mM 0.5457 mL 2.7285 mL 5.4570 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molaritätsrechner

  • Verdünnungsrechner

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Reinheit & Dokumentation

Purity: 98.80%

SDS (251 KB)

COA (249 KB)

Handling Instructions (2659 KB)
Verweise

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.7285 mL 13.6426 mL 27.2851 mL 68.2128 mL
5 mM 0.5457 mL 2.7285 mL 5.4570 mL 13.6426 mL
10 mM 0.2729 mL 1.3643 mL 2.7285 mL 6.8213 mL
15 mM 0.1819 mL 0.9095 mL 1.8190 mL 4.5475 mL
20 mM 0.1364 mL 0.6821 mL 1.3643 mL 3.4106 mL
25 mM 0.1091 mL 0.5457 mL 1.0914 mL 2.7285 mL
30 mM 0.0910 mL 0.4548 mL 0.9095 mL 2.2738 mL
40 mM 0.0682 mL 0.3411 mL 0.6821 mL 1.7053 mL
50 mM 0.0546 mL 0.2729 mL 0.5457 mL 1.3643 mL
60 mM 0.0455 mL 0.2274 mL 0.4548 mL 1.1369 mL
80 mM 0.0341 mL 0.1705 mL 0.3411 mL 0.8527 mL
100 mM 0.0273 mL 0.1364 mL 0.2729 mL 0.6821 mL
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RXR antagonist 5 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

RXR antagonist 51807740-94-8RXR antagonist5RXR antagonist-5RAR/RXRRetinoic acid receptorsRetinoid X receptorsInhibitorinhibitorinhibit

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