2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. Talibegron hydrochloride

Talibegron hydrochloride  (Synonyms: ZD2079 hydrochloride)

製品番号: HY-15378 純度: 99.63%
COA 取扱説明書 Technical Support

Talibegron hydrochloride (ZD2079 hydrochloride) is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Talibegron hydrochloride has potent vasorelaxant effect.

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Talibegron hydrochloride

Talibegron hydrochloride 構造式

CAS 番号 : 178600-17-4

容量 価格（税別） 在庫状況 数量
1 mg $30 在庫あり
5 mg $75 在庫あり
10 mg $120 在庫あり
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100 mg   お問い合わせ  

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Talibegron hydrochloride 関連抗体

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製品説明

Talibegron hydrochloride (ZD2079 hydrochloride) is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Talibegron hydrochloride has potent vasorelaxant effect[1].

体外実験

Talibegron hydrochloride (ZD2079 hydrochloride; 0.01-1000 μM) produces a concentration-dependent relaxation of phenylephrine-preconstricted isolated mesenteric arteries and causes full relaxation with 1 mM[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Talibegron hydrochloride 関連抗体
分子量

351.82

分子式

C18H22ClNO4
CAS 番号
Appearance

Solid

Color

White to off-white

SMILES

O=C(O)CC1=CC=C(OCCNC[C@H](O)C2=CC=CC=C2)C=C1.[H]Cl
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
溶剤 & 溶解度
体外: 

DMSO : 125 mg/mL (355.30 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.8424 mL 14.2118 mL 28.4236 mL
5 mM 0.5685 mL 2.8424 mL 5.6847 mL
10 mM 0.2842 mL 1.4212 mL 2.8424 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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一般には略語で表示されます：C1V1 = C2V2

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純度とドキュメンテーション
参考文献

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.8424 mL 14.2118 mL 28.4236 mL 71.0591 mL
5 mM 0.5685 mL 2.8424 mL 5.6847 mL 14.2118 mL
10 mM 0.2842 mL 1.4212 mL 2.8424 mL 7.1059 mL
15 mM 0.1895 mL 0.9475 mL 1.8949 mL 4.7373 mL
20 mM 0.1421 mL 0.7106 mL 1.4212 mL 3.5530 mL
25 mM 0.1137 mL 0.5685 mL 1.1369 mL 2.8424 mL
30 mM 0.0947 mL 0.4737 mL 0.9475 mL 2.3686 mL
40 mM 0.0711 mL 0.3553 mL 0.7106 mL 1.7765 mL
50 mM 0.0568 mL 0.2842 mL 0.5685 mL 1.4212 mL
60 mM 0.0474 mL 0.2369 mL 0.4737 mL 1.1843 mL
80 mM 0.0355 mL 0.1776 mL 0.3553 mL 0.8882 mL
100 mM 0.0284 mL 0.1421 mL 0.2842 mL 0.7106 mL
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Talibegron hydrochloride Related Classifications

  • Molarity Calculator

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

質量   濃度   体積   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

一般には略語で表示されます：C1V1 = C2V2

濃度 （開始） × 体積 （開始） = 濃度 （終了） × 体積 （終了）
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Talibegron178600-17-4ZD2079ZD 2079ZD-2079Adrenergic ReceptorBeta Receptorβ3adrenoceptorpD2phenylephrinepreconstrictedmesentericarteryvasorelaxantInhibitorinhibitorinhibit

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製品名:
Talibegron hydrochloride
製品番号:
HY-15378
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