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Ipenoxazone (Synonyms: MLV-6976; NC-1200)

Cat. No.: HY-100159
Handling Instructions

Ipenoxazone is a potent and centrally acting muscle relaxant.

For research use only. We do not sell to patients.

Ipenoxazone Chemical Structure

Ipenoxazone Chemical Structure

CAS No. : 104454-71-9

Size Price Stock
1 mg USD 1502 Get quote
5 mg USD 2404 Get quote
10 mg USD 3847 Get quote

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Customer Review

  • Biological Activity

  • Protocol

  • Technical Information

  • Purity & Documentation

  • References

Description

Ipenoxazone is a potent and centrally acting muscle relaxant.

In Vivo

Ipenoxazone is a potent and centrally acting muscle relaxant[1]. An intravenous injection of 2 mg/kg Ipenoxazone causes a reduction of electromyographic activity which reaches a maximum within 3 min after the injection. Within 1 min after the injection of Ipenoxazone at a dose of 4 mg/kg, the blood pressure changes from a control level of 138±9 mmHg to a minimum level of 98±9 mmHg (n=6) but it rapidly returns to the control level within 1 to 2 min, while the rigidity is still reduced significantly at that time. High doses (greater than 30 mg/kg i.p.) of Ipenoxazone produces a transient and dose-dependent sedation in almost all mice about 5 min after its administration[2].

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.7892 mL 13.9462 mL 27.8924 mL
5 mM 0.5578 mL 2.7892 mL 5.5785 mL
10 mM 0.2789 mL 1.3946 mL 2.7892 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Animal Administration
[1]

Experiments are performed on 31 adult male rats (Wistar 310 to 430 g, 3 to 7 months of age) anesthetized with chloralose-urethane (50 and 500 mg/kg i.p., respectively). Ipenoxazone is administrated i.v. at 0.05 to 0.1 mL/100 g body weight (20 to 40 s per injection). These four different doses of Ipenoxazone (0.3, 1, 3 and 10 mg/kg) are administrated cumulatively, from small doses to larger doses. It is usually waited about 10 to 30 min between each trial or until all effects of the drug on the bladder have disappeared[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

References
Molecular Weight

358.52

Formula

C₂₂H₃₄N₂O₂

CAS No.

104454-71-9

SMILES

O=C1O[[email protected]](C2=CC=CC=C2)[[email protected]](CC(C)C)N1CCCN3CCCCCC3

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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Product Name:
Ipenoxazone
Cat. No.:
HY-100159
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Ipenoxazone

Cat. No.: HY-100159