2. Signaling Pathways
  3. GPCR/G Protein
  4. Prostaglandin Receptor
  5. EP Isoform
  6. EP Inhibitor

EP Inhibitor

EP Inhibitors (7):

Cat. No. Product Name Effect Purity
  • HY-100441
    Treprostinil
    		Inhibitor 99.98%
    Treprostinil (UT-15) is a potent DP1 and EP2 agonist with EC50 values of 0.6±0.1 and 6.2±1.2 nM, respectively.
  • HY-108559
    L-161982
    		Inhibitor 99.04%
    L-161982 is a selective EP4 receptor antagonist.
  • HY-N0314
    Pectolinarin
    		Inhibitor 99.89%
    Pectolinarin possesses anti-inflammatory activity.
  • HY-136895
    AZ12672857
    		Inhibitor 98.44%
    AZ12672857 is an orally active inhibitor of EphB4 (IC50=1.3 nM) and Src kinases.
  • HY-N0223
    Epibetulinic acid
    		Inhibitor ≥98.0%
    Epibetulinic acid exhibits potent inhibitory effects on NO and prostaglandin E2 (PGE2) production in mouse macrophages (RAW 264.7) stimulated with bacterial endotoxin with IC50s of 0.7 and 0.6 μM, respectively.
  • HY-138761
    EP4 receptor antagonist 3
    		Inhibitor
    EP4 receptor antagonist 3 is a potent EP4 receptor antagonist, example 3,extracted from patent WO2010019796 A1.
  • HY-N2569
    (-)-Curine
    		Inhibitor
    (-)-Curine is an orally active bisbenzylisoquinoline alkaloid isolated from Chondrodendron platyphyllum.