Alimemazine (Synonyms: Trimeprazine)

Art. -Nr.: HY-12752: Data Sheet Handling Instructions
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Alimemazine is a phenothiazine derivative that is generally used as an antipruritic agent and also a hemagglutinin (HA)-receptor antagonist.Alimemazine (Trimeprazine) is also acts as a partial agonist against the histamine H1 receptor (H1R) and other GPCRs. Alimemazine displays antiserotonin, antispasmodic, and antiemetic properties.

At equivalent molar concentrations, both the salt and free forms of a compound exhibit comparable biological activity. Nevertheless, the salt form (Alimemazine hemitartrate) usually boasts enhanced water solubility and stability.

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Alimemazine Chemische Struktur

CAS. Nr. : 84-96-8

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Other In-stock Forms of Alimemazine:

Alimemazine hemitartrate

Other Forms of Alimemazine:

Alimemazine-d₆ In-stock
Alimemazine hemitartrate In-stock
Alimemazine-d₆ hydrochloride Angebot einholen

Spezialitätsempfehlungen

•Related Small Molecules:

•Related Proteins:

Alle Histamine Receptor Isoform-spezifische Produkte anzeigen:

Alle Isoformen anzeigen

H₁ Receptor H₂ Receptor H₃ Receptor H₄ Receptor Histamine Receptor

Biologische Aktivität
Reinheit & Dokumentation
Verweise
Kundenbewertung

Beschreibung

IC₅₀ & Target

H₁ Receptor

Molekulargewicht

298.45

Formel

C₁₈H₂₂N₂S

CAS. Nr.

84-96-8

SMILES

CC(CN(C)C)CN1C2=CC=CC=C2SC3=CC=CC=C31

Versand

Room temperature in continental US; may vary elsewhere.

Speicherung

Please store the product under the recommended conditions in the Certificate of Analysis.

Reinheit & Dokumentation

Handling Instructions (2659 KB)

Verweise

[1]. Singh B, et al. Bioanalytical method development and validation of alimemazine in human plasma by LC-MS/MS and its application in bioequivalence studies. J Pharm Bioallied Sci. 2013 Oct;5(4):257-64. [Content Brief]

[2]. Kuznetsova A, et al. Trimeprazine increases IRS2 in human islets and promotes pancreatic β cell growth and function in mice. JCI Insight. 2016;1(3). [Content Brief]

Alimemazine Related Classifications

Molaritätsrechner
Verdünnungsrechner

Die Formel zur Berechnung von Molaritäten

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass		Concentration		Volume		Molecular Weight *
	=		×		×

The dilution calculator equation

Konzentration _{(Stammlösung)} × Volumen _{(Stammlösung)} = Konzentration _{(Ziellösung)} × Volumen _{(Ziellösung)}

Diese Gleichung wird häufig abgekürzt als: C₁V₁ = C₂V₂

Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Alimemazine84-96-8TrimeprazineHistamine Receptorhemagglutininhistamin-H1Inhibitorinhibitorinhibit

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