2. GPCR/G Protein
  3. Protease Activated Receptor (PAR)
  4. FSLLRY-NH2

FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor.

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Custom Peptide Synthesis

FSLLRY-NH2

FSLLRY-NH2 화학구조

CAS No. : 245329-02-6

사이즈 가격 재고 수량
1 mg 해외재고보유
5 mg 해외재고보유
10 mg 해외재고보유
25 mg 해외재고보유
50 mg   견적 받기  
100 mg   견적 받기  

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

This product is a controlled substance and not for sale in your territory.

고객리뷰

Based on 6 publication(s) in Google Scholar

Other Forms of FSLLRY-NH2:

FSLLRY-NH2 Related Antibodies

Top Publications Citing Use of Products

View All Protease Activated Receptor (PAR) Isoform Specific Products:

View All Isoforms
PAR1 PAR2 PAR4

  • Biological Activity

  • 순도&문서

  • References

  • 고객리뷰

제품 설명

FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor[1].

IC50 & Target

PAR2

 

In Vivo

Treatment with FSLLRY-NH2 (50 μg per rat administered intranasally at 1 hour postresuscitation) significantly improves neurological outcome and reduces the number of degenerating hippocampal neurons after ACA (asphyxial CA)[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
분자량

796.96

화학식

C39H60N10O8
CAS No.
Appearance

Solid

Color

White to off-white

Sequence

Phe-Ser-Leu-Leu-Arg-Tyr-NH2
Sequence Shortening

FSLLRY-NH2
선적

Room temperature in continental US; may vary elsewhere.
보관

Sealed storage, away from moisture and light

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

용액&용해도
In Vitro: 

DMSO : 100 mg/mL (125.48 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.2548 mL 6.2738 mL 12.5477 mL
5 mM 0.2510 mL 1.2548 mL 2.5095 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • 몰농도 계산기

  • 농도 희석 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
순도&문서
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 1.2548 mL 6.2738 mL 12.5477 mL 31.3692 mL
5 mM 0.2510 mL 1.2548 mL 2.5095 mL 6.2738 mL
10 mM 0.1255 mL 0.6274 mL 1.2548 mL 3.1369 mL
15 mM 0.0837 mL 0.4183 mL 0.8365 mL 2.0913 mL
20 mM 0.0627 mL 0.3137 mL 0.6274 mL 1.5685 mL
25 mM 0.0502 mL 0.2510 mL 0.5019 mL 1.2548 mL
30 mM 0.0418 mL 0.2091 mL 0.4183 mL 1.0456 mL
40 mM 0.0314 mL 0.1568 mL 0.3137 mL 0.7842 mL
50 mM 0.0251 mL 0.1255 mL 0.2510 mL 0.6274 mL
60 mM 0.0209 mL 0.1046 mL 0.2091 mL 0.5228 mL
80 mM 0.0157 mL 0.0784 mL 0.1568 mL 0.3921 mL
100 mM 0.0125 mL 0.0627 mL 0.1255 mL 0.3137 mL
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FSLLRY-NH2 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

FSLLRY-NH2245329-02-6Protease Activated Receptor (PAR)Thrombin receptorsInhibitorinhibitorinhibit

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Inquiry Information

상품명:
FSLLRY-NH2
Cat. No.:
HY-P1260
수량:
MCE Japan Authorized Agent:

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비고

SAFETY DATA SHEET (SDS)

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