1. GPCR/G Protein
  2. Protease-Activated Receptor (PAR)
  3. FSLLRY-NH2 TFA

FSLLRY-NH2 TFA 

Cat. No.: HY-P1260A Purity: 98.20%
Handling Instructions

FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

FSLLRY-NH2 TFA Chemical Structure

FSLLRY-NH2 TFA Chemical Structure

Size Price Stock Quantity
5 mg USD 190 In-stock
Estimated Time of Arrival: December 31
10 mg   Get quote  
50 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of FSLLRY-NH2 TFA:

Top Publications Citing Use of Products
  • Biological Activity

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Description

FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor[1].

In Vivo

Treatment with FSLLRY-NH2 (50 μg per rat administered intranasally at 1 hour postresuscitation) significantly improves neurological outcome and reduces the number of degenerating hippocampal neurons after ACA (asphyxial CA)[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

910.98

Formula

C₄₁H₆₁F₃N₁₀O₁₀

Sequence

Phe-Ser-Leu-Leu-Arg-Tyr-NH2

Sequence Shortening

FSLLRY-NH2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -80°C 2 years
-20°C 1 year
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (109.77 mM; Need ultrasonic)

H2O : 1.43 mg/mL (1.57 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.0977 mL 5.4886 mL 10.9772 mL
5 mM 0.2195 mL 1.0977 mL 2.1954 mL
10 mM 0.1098 mL 0.5489 mL 1.0977 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (2.74 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (2.74 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (2.74 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

FSLLRY-NH2Protease-Activated Receptor (PAR)Thrombin receptorsInhibitorinhibitorinhibit

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Product Name:
FSLLRY-NH2 TFA
Cat. No.:
HY-P1260A
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