2. Vitamin D Related/Nuclear Receptor
  3. Estrogen Receptor/ERR
  4. GPR30 agonist-1

GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects.

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GPR30 agonist-1

GPR30 agonist-1 構造式

CAS 番号 : 415919-74-3

容量 価格（税別） 在庫状況 数量
>無料サンプル (0.1 - 0.2 mg)   今すぐ申し込む  
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO
ready for reconstitution
 USD 132 在庫あり
Solution
10 mM * 1 mL in DMSO USD 132 在庫あり
Solid
5 mg $120 在庫あり
10 mg $200 在庫あり
25 mg $390 在庫あり
50 mg $600 在庫あり
100 mg   お問い合わせ  
200 mg   お問い合わせ  

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GPR30 agonist-1 関連抗体

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Estrogen receptor ERα ERβ ERRα ERRβ ERRγ

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製品説明

GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects[1].

体内実験

GPR30 agonist-1 (compound 5408-0877) (1 nM-10 μM) induces a concentration-dependent relaxation in carotid arteries from both male and female rats. GPR30 agonist-1-induced relaxation is abolished by endothelium removal and abrogated in the presence of the nitric oxide synthase inhibitor NG-nitro-l-arginine methyl ester (100 μM)[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

374.25

分子式

C19H17BrFNO
CAS 番号
Appearance

Solid

Color

White to off-white

SMILES

COC(C=C1)=C(C=C1Br)[C@@]2([H])[C@](CC=C3)([H])[C@]3([H])C4=CC(F)=CC=C4N2
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
溶剤 & 溶解度
体外: 

DMSO : 50 mg/mL (133.60 mM; ultrasonic and warming and heat to 80°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6720 mL 13.3601 mL 26.7201 mL
5 mM 0.5344 mL 2.6720 mL 5.3440 mL
10 mM 0.2672 mL 1.3360 mL 2.6720 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

一般には略語で表示されます：C1V1 = C2V2

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体積 （開始）

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In Vivo Dissolution Calculator
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純度とドキュメンテーション
参考文献

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.6720 mL 13.3601 mL 26.7201 mL 66.8003 mL
5 mM 0.5344 mL 2.6720 mL 5.3440 mL 13.3601 mL
10 mM 0.2672 mL 1.3360 mL 2.6720 mL 6.6800 mL
15 mM 0.1781 mL 0.8907 mL 1.7813 mL 4.4534 mL
20 mM 0.1336 mL 0.6680 mL 1.3360 mL 3.3400 mL
25 mM 0.1069 mL 0.5344 mL 1.0688 mL 2.6720 mL
30 mM 0.0891 mL 0.4453 mL 0.8907 mL 2.2267 mL
40 mM 0.0668 mL 0.3340 mL 0.6680 mL 1.6700 mL
50 mM 0.0534 mL 0.2672 mL 0.5344 mL 1.3360 mL
60 mM 0.0445 mL 0.2227 mL 0.4453 mL 1.1133 mL
80 mM 0.0334 mL 0.1670 mL 0.3340 mL 0.8350 mL
100 mM 0.0267 mL 0.1336 mL 0.2672 mL 0.6680 mL
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GPR30 agonist-1 Related Classifications

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

質量   濃度   体積   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

一般には略語で表示されます：C1V1 = C2V2

濃度 （開始） × 体積 （開始） = 濃度 （終了） × 体積 （終了）
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPR30 agonist-1415919-74-3Estrogen Receptor/ERRGPR30vasorelaxantestrogenInhibitorinhibitorinhibit

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製品名:
GPR30 agonist-1
製品番号:
HY-138686
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